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1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-hydroxy-N-[3-(pyridin-2-yl)propyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2,4-dimethyl-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]pyrimidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-(4-fluorophenyl)-2-hydroxy-N-[3-(pyridin-4-yl)propyl]acetamide
4-[(quinoxalin-2-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
1-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]-2-phenylethan-1-ol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)methyl]phenol
(2S)-2-hydroxy-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]butanoic acid
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(pyridin-3-ylmethyl)urea
(5S,9aS,9bS)-2-cyclopentyl-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-(pyridin-2-yl)acetamide
N-[4-(propan-2-yl)phenyl]-1-(pyridin-3-ylmethyl)piperidin-3-amine
3-[(6-methoxypyrimidin-4-yl)(methyl)amino]-1-phenylpropan-1-ol
1-methyl-3-phenyl-4-(quinoxalin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-{2-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]ethyl}benzoic acid
N-[2-(1H-imidazol-4-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
{1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2-cyclopropylpyrimidin-5-yl)-N-ethyl-7-methoxy-N-methylquinoline-4-carboxamide
1-(4-methoxyphenyl)-6,6-dimethyl-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1R,5R)-6-methyl-3-[2-(trifluoromethoxy)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
3-{2-[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(2-methoxyphenyl)ethyl]-2-(4-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
9-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
N-[(3R,4S)-1-cyclopentanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
8-(5,6-dimethylpyrimidin-4-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenoxybutanamide
1-(3-cyano-4-methylphenyl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]urea
N-[2-(1H-indol-3-yl)ethyl]-2,6-dimethyl-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
methyl 3-[(furan-3-ylformamido)methyl]-5-(2-methoxybenzamido)benzoate
3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(morpholin-4-yl)propan-1-one
4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
N-[4-({[(2R)-1-hydroxy-3-methylbutan-2-yl]carbamoyl}methyl)phenyl]butanamide
N-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
N-(isoquinolin-5-ylmethyl)-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-N-(2-phenylethyl)-N-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-amine
2-[5-(1-ethylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
6-oxo-1-(2-phenylethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]piperidine-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethan-1-one
4-[3-(azocane-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-[2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
4-(benzyloxy)-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine
3-(2-methoxyphenyl)-N-[1-({[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide