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2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
7-(2-methoxyethyl)-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{2-[4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-{1-[2-(1,4-dimethylpiperazin-2-yl)acetyl]piperidin-4-yl}-N-phenylpropanamide
3-[(dimethylamino)methyl]-1-(4-propylpyrimidine-5-carbonyl)piperidin-3-ol
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxybutan-1-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-(thiophen-3-ylmethyl)urea
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
5-ethyl-N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[(4-phenylmorpholin-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-methylquinoline
3-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
1-cyclopentanecarbonyl-N-[2-(5-methylthiophen-2-yl)ethyl]piperidine-4-carboxamide
4-(1H-imidazol-1-yl)-1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidine-4-carboxylic acid
9-hydroxy-N-methyl-4-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoline
N,2-diethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-4-(4-methylpiperazin-1-yl)pentan-1-one
(3S,4S)-1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
ethyl 1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
4-methoxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
methyl 3-{[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
(3S,9aR)-3-(4-aminobutyl)-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-1-(1-benzothiophen-2-ylmethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-ethoxy-1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
N-methyl-N-[(6-methylquinolin-5-yl)methyl]oxan-4-amine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetamide
2-{[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl](methyl)amino}-N-methylacetamide
2-(4-{[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
1-{1'-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-cyclopentyl-4-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]-4-oxobutanamide
3-[2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamido]-N-methylpropanamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-N,N-dimethyl-2-oxo-decahydro-1,6-naphthyridine-6-sulfonamide
1-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]cyclopropane-1-carboxamide
4-ethyl-N,N-dimethyl-6-(4-{[2-(pyridin-3-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
(3S,4S)-4-cyclopropyl-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}pyrrolidine-3-carboxylic acid
5-(3-chlorophenyl)-3-[4-(pyrimidin-2-yl)piperazin-1-yl]-1,2,4-triazine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-hydroxy-N,2-dimethylbenzamide
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
(1R,5R)-3-(3-chloro-4-fluorobenzoyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-(2-methylphenyl)-1,3-thiazole
5-ethyl-N4-methyl-N4-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidine-2,4-diamine
4-(2-cyanophenyl)-N-propylbenzamide
N-methyl-1-[(4-methylphenyl)amino]-N-[1-(1,3-thiazol-2-yl)ethyl]cyclopentane-1-carboxamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-[4-(furan-2-yl)phenyl]-1H-imidazole
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-phenyl-1,4-diazepane-1-carboxamide
N-cyclopropyl-2-(quinoxalin-6-ylformamido)acetamide