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2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
[(3R,4R)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1λ6-thiomorpholine-1,1-dione
3-[1-(4-methoxybenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-[9-(4-cyanobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)acetamide
methyl 2-[3-oxo-1-(1H-1,2,4-triazole-5-carbonyl)piperazin-2-yl]acetate
N-{2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
2-[methyl(2-phenylethyl)amino]-N-(oxan-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
3-{[2-(dimethylamino)ethyl]({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)carbamoyl}pyridin-1-ium-1-olate
2-(4-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-(2,3-dihydro-1H-inden-2-yl)-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
2-ethyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,3,4-thiadiazole
N-cyclopropyl-N-{[1-(pent-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
5-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-N-ethyl-4-methyl-1,3-thiazol-2-amine
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
4-[2-(4-chlorophenyl)morpholin-4-yl]butan-1-ol
1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[1-(2-phenylethyl)piperidin-3-yl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
6-(2-methyl-1,3-thiazol-4-yl)-2-[2-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(3-methylphenyl)methyl]-4-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperazin-2-one
(5S,9aS,9bS)-5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-chloro-5-(7-methyl-1H-indol-3-yl)benzamide
2-{1-[(4-fluorophenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}dimethylamine
(1R,7S)-6-(3-oxo-1,4-diazepane-1-carbonyl)-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(3-methoxyphenyl)methyl]-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,7aR)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropanecarbonyl-8-(4-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-dimethyl-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazine-1-carboxamide
3-[5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
3-(3-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propoxy)pyridine
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
3-(pyrrolidine-1-carbonyl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]piperidine
N-methyl-2-{[(3-methylthiophen-2-yl)methyl]amino}-N-(1H-pyrazol-5-ylmethyl)benzamide
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2,6,8-trimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
3-(3,4-dimethylphenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
(1S,5R)-6-(2-methoxyethyl)-3-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-N-methyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(1H-indol-3-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide