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1-[3-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(3-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}phenyl)-3,5-dimethyl-1H-pyrazole
4-(4-benzyl-1H-pyrazol-5-yl)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidine
3-amino-1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}pyrrolidine-3-carboxylic acid
ethyl 1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
3-{[(3-methyl-1,2-oxazol-5-yl)methyl]sulfamoyl}-N-(pyridin-2-ylmethyl)benzamide
3-[(2-hydroxyethyl)({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
1-({1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
(2S,4S)-N-ethyl-1-(furan-2-ylmethyl)-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
6-(dimethylamino)-N-[2-(2-methylpropanesulfonyl)ethyl]pyridine-3-carboxamide
1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
5-ethyl-2-methyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-(quinoxalin-6-ylmethyl)piperidine-3-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
5-[(5-phenylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-benzyl-N3-ethyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
3-[3-(methoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-[1-(6-chloropyridazin-3-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(1-{3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-methoxyacetamide
6-{[butyl(methyl)amino]methyl}-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]azetidin-3-yl}pyridine
2-methoxy-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-(quinoxalin-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
2-{1-[6-(propan-2-yl)-1H-indole-2-carbonyl]piperidin-3-yl}ethan-1-amine
1-[2-(morpholin-4-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
N-methyl-2-(pyrrolidin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
7-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[1-(2-hydroxypropyl)-1H-imidazol-2-yl]benzamide
(3S,4R)-1-(2-amino-9H-purin-6-yl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1-[2-(methylsulfanyl)benzoyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
benzyl({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})ethylamine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamide
1-(furan-3-ylmethyl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid
2-(2-methyl-1,3-benzothiazol-5-yl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N3-cyclooctyl-N5-(1-methoxybutan-2-yl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-methyl-2-(pyrrolidin-1-yl)propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-N-methyloxolan-3-amine
(1-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
5-acetyl-N,2,4-trimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrrole-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(2-methylpropyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide