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N-[2-(3-chlorophenyl)ethyl]-2-[2-(pyridin-2-yl)piperidin-1-yl]acetamide
2-methoxy-N-{1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
6-{4-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N,2,6-trimethyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)quinoline-4-carboxamide
6-fluoro-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-benzyl-N-methyl-3-({[(5-phenyl-1H-pyrazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(4-propylpyrimidine-5-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}[2-(3-fluorophenyl)ethyl]amine
1-methyl-6-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2-methoxyethyl)[2-phenyl-1-(1-propylpiperidin-4-yl)ethyl](pyridin-2-ylmethyl)amine
3-{2-amino-4-methyl-6-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidin-5-yl}propanoic acid
7-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}quinolin-8-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxybutanamide
methyl (2S,4S)-4-acetamido-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxylate
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-phenylprop-2-yn-1-one
5-[methyl(2-phenylethyl)amino]-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-4-{[4-(morpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
7-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
4,6-dimethyl-1-{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
1,3-dimethyl-2,6-dioxo-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl 1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(2-methoxyphenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-(furan-3-ylmethyl)-4-(4-methoxyphenoxy)benzamide
2-amino-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
3-(2-chlorophenyl)-3-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1-methylpyrrolidine-2,5-dione
8-methoxy-2-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinoline
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine
1-{6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
1-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
1-[2-(hydroxymethyl)azepan-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
[(3R,4R)-1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
{4-benzyl-1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methanol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(4-methylpiperazin-1-yl)benzamide
(2S,4R)-4-[4-chloro-3-(1H-pyrrol-1-yl)benzamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
2-(4-chloro-2-methylphenoxy)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[3-(4-methoxyphenyl)propyl]-6-[(1-methylpiperidin-3-yl)amino]pyridine-3-carboxamide
(1S,5R)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(4-methyl-1H-imidazol-5-yl)methyl](oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
6-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine
8-(2-butoxyacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-[4-(3,4-difluorobenzoyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine