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6-methoxy-N-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,3-benzothiazol-2-amine
4-({1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)morpholine
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-ethyl-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-benzyl-4-[2-(1H-imidazol-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
2-(4-{[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclohexyl)-1H-1,3-benzodiazole
4-(2-methylphenoxy)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-[4-(1H-1,3-benzodiazol-6-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-[4-(2,2-dimethylmorpholin-4-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
3-(3-{[(1H-imidazol-2-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide
2-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-4-(2-oxopyrrolidin-1-yl)benzamide
2-cyclopropyl-N-[2-(methylsulfanyl)ethyl]-1,3-benzoxazole-6-carboxamide
8-(1,4-dioxan-2-ylmethyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({[(3R,4R)-1-[(3,4-difluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-amino-6-cyclopropyl-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
4-[3-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-ethyl-5-methyl-1,2-oxazole
5,6-dimethyl-3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(azocan-1-yl)-3-[4-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-3-propylpiperidin-3-yl)methanol
1-(4-aminobutanoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(ethanesulfonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,4R)-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-N,N-diethylpyrrolidine-2-carboxamide
2-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-({4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-3,4-dihydroquinazolin-4-one
4-(5-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(thiophen-2-yl)propanamide
7-[2-(3-methylphenyl)benzoyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
1-methyl-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
1-ethyl-3-(hydroxymethyl)-N-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
8-benzyl-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(azetidine-1-sulfonyl)-N-[2-(2-fluorophenyl)ethyl]benzamide
(3R,4R)-4-(azepan-1-yl)-1-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-ol
8-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dihydro-1H-inden-2-yl)-N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
2-amino-6-{4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[5-(2-methyl-4-phenylpyridin-3-yl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-3-(methoxymethyl)piperidine
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}pyridine-2-carboxamide
(2S,4R)-4-amino-1-(3-hydroxy-2-methylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(1-{2-[3-(benzyloxy)phenyl]-1H-imidazol-1-yl}ethyl)-4-methyl-4H-1,2,4-triazole
1-cyclopropanecarbonyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
1-(4-cyclohexylphenyl)-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
methyl 4-(5-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide