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5-methoxy-1-methyl-N-[3-(phenylsulfanyl)propyl]-1H-indole-2-carboxamide
N-tert-butyl-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
[5-(4-cyclopentylpyrimidin-2-yl)-2-fluorophenyl]methanol
1-(2-chlorophenyl)-5-methyl-4-(quinoline-6-carbonyl)piperazin-2-one
1-cyclopropanecarbonyl-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
2-methyl-N-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)propanamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-hydroxypyridine-2-carboxamide
3,5-dimethyl-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl}-1H-pyrazole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-methyl-5-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}pyrimidin-2-amine
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
1-{3-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
2-{2-[1-(2-propoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
3-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1-[2-(4-methoxyphenyl)phenyl]urea
N-[2-(1,3-benzothiazol-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-N-(2-methylpropyl)-2-oxoacetamide
2-(4-methoxyphenyl)-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[4-(pyrimidin-2-yl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-(2-ethylbutyl)-8-(3-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(1R,5R)-3-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-N-ethylacetamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-ol
2-[1-(cyclohexylmethyl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpiperidin-3-amine
ethyl 4-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine
1-[1-(3-hydroxy-4-methylbenzoyl)piperidin-4-yl]pyrrolidin-2-one
4-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
1-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-cyclopropanecarbonyl-1'-(2,2-dimethyloxane-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[3-(2-ethoxyphenyl)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
1-[(4-chlorophenyl)methyl]-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
2-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}-4-methyl-1,3-thiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-ol
1-[5-(4-methanesulfonylpiperazine-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]pyrimidine
(3S,4S)-3-hydroxy-4-(morpholin-4-yl)-N-(3-phenylphenyl)pyrrolidine-1-carboxamide
methyl 3-(5-methyl-1,2-oxazole-3-carbonyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{2-[1-(4-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
4-(2H-1,3-benzodioxol-5-yl)-3-butyl-1-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,7S)-3-(2-acetamidoethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl[2-(1H-pyrazol-1-yl)ethyl]{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine