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dimethyl({5-[4-(1H-1,2,4-triazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)amine
2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyrimidin-4-amine
N-(adamantan-2-ylmethyl)-6-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(dimethyl-1,3-thiazol-4-yl)-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]acetamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
4-ethyl-3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
8-[3-(2-oxopyrrolidin-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-oxo-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(3S,4S)-3-hydroxy-N-[3-(2-oxopyrrolidin-1-yl)phenyl]-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
6-phenyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyridine-3-carboxylic acid
5-chloro-2-(morpholine-4-carbonyl)-3-phenyl-1H-indole
3,5-dimethyl-1-(3-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propyl)-1H-pyrazole
{2-[(5-chloropyridin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
2-[2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-(4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
N-cyclopropyl-2-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}pyridine-4-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-methyl-2-(oxolane-3-carbonyl)-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
methyl 2-[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)(methyl)amino]acetate
N-[1-(4-fluorophenyl)-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-methyl-1,3-thiazole-5-carboxamide
3-(propan-2-yl)-1-{[1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methyl}urea
4-hydroxy-N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-methylbenzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(2R,3R,6R)-5-(2-ethoxypyridine-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(2-fluorophenyl)-3-[4-(2-phenoxyethyl)piperazin-1-yl]-1,2,4-triazine
N-benzyl-1-(2-hydroxyethyl)-5-[(3-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
3-{5-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)-1,3-thiazole
(2S,4S)-1-benzyl-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine
N-[(5-methyl-2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2-hydroxyethyl)-N-methyl-1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N,2-dimethyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-(4H-1,2,4-triazol-4-yl)pyridine
11-{[3-(methylsulfanyl)propyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
N-(4-{3H-imidazo[4,5-b]pyridin-5-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)piperidin-4-amine
4,6-dimethyl-1-{3-oxo-3-[2-(trifluoromethyl)pyrrolidin-1-yl]propyl}-1,2-dihydropyrimidin-2-one
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-[3-(methylsulfanyl)phenyl]acetamide
3-methyl-N-(2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
(1R,5R)-6-[2-(1H-indol-3-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide