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6-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carbonitrile
1-[bis(4-fluorophenyl)methyl]-4-(1H-imidazol-4-ylmethyl)piperazine
(4aS,8aR)-6-(2-methoxy-2-methylpropanoyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-4-ol
7-(cyclohexylmethyl)-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
N-cyclopentyl-5-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrazine-2-carboxamide
6-(4-methoxyphenyl)-9-(1H-pyrazol-3-ylmethyl)-6,9-diazaspiro[4.5]decan-7-one
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(3R,4R)-1-(dimethyl-1,3-thiazol-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N,N-dimethyl-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}aniline
N-{[4-(methylsulfanyl)phenyl]methyl}-N-propylbutanamide
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
2-methyl-4-(4-{[4-(thian-4-yl)piperazin-1-yl]methyl}phenyl)butan-2-ol
N3-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(4-fluorophenoxy)-1-(oxolan-3-ylmethyl)piperidine
N-[2-(4-methoxyphenyl)ethyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
2-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-2-yl}ethan-1-ol
3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
methyl 4-(4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)benzoate
{2-[2-benzyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}urea
8-{[3-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,4-diazepane-6-carboxylic acid
{4-[(2,3-dimethyl-1H-indol-7-yl)methyl]morpholin-3-yl}methanol
3-acetyl-N-[(1-benzylpyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-(morpholin-4-yl)butanamide
1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-(4-fluorophenyl)ethan-1-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-oxo-2H-chromene-3-carboxamide
2-(3,4-dichlorophenyl)-4-(2-propoxyethyl)morpholine
7-(1,3-benzothiazol-2-yl)-4-(1,4-dioxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(4-chlorophenyl)-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclopropane-1-carboxamide
4-(5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
2-(methylamino)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyridine-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(1,2-oxazolidin-2-yl)propanamide
1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
8-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(2-amino-1,3-thiazol-4-yl)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]propan-1-one
2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-3,5-dimethoxybenzoic acid
4-({2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-1,3-dimethylpiperazin-2-one
6-methoxy-2-oxo-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(1H-imidazol-2-yl)piperidine
(1R,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[1-(cyclopropylmethyl)piperidin-3-yl]ethyl}pyridine-4-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-ol