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5,6-dimethyl-2-[4-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-methyl-4-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
2-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-[3-(cyclopropylmethyl)-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]propan-1-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
2-chloro-5-(3,5-dimethyl-1H-pyrazol-4-yl)benzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
4-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-1,3-thiazole-5-carboxamide
1-(3-fluorophenyl)-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
8-(3-methylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methoxy-1-[1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-methyl-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}butanamide
N-[4-(1-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
3-[2-(ethanesulfonyl)ethyl]-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
ethyl 5-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-[1-(3-ethoxypropyl)-1H-imidazol-2-yl]pyridine
2-({4-[5-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
1-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
3-ethyl-5-hydroxy-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]adamantane-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-3-ol
4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
3-(4-chlorobenzoyl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
2,6-dimethyl-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]pyrimidin-2-amine
2-{1-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-imidazol-2-yl}pyridine
1-cyclohexanecarbonyl-4-(5-propyl-1,2-oxazole-3-carbonyl)piperazine
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
6-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[3-(3-methoxyphenyl)phenyl]-1-[3-(morpholin-4-yl)propyl]urea
3-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{1-[(4-ethoxyphenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-[2-(5-methylfuran-2-yl)ethyl]-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
[(5-chlorothiophen-2-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
N-[2-(2-hydroxyethoxy)ethyl]-2,3-dihydro-1H-indene-1-carboxamide
2-(1-benzyl-5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,4-triazol-3-yl)acetamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-phenylethan-1-one
4-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-hydroxyphenyl)ethan-1-one
4-(5-methylpyridin-2-yl)-1-(quinoline-6-carbonyl)piperidin-4-ol
1-(furan-2-ylmethyl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]piperidine-3-carboxamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(9aR)-2-methyl-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-chloro-1,3-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(5-acetylthiophen-3-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}propan-1-one
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-2-methyl-1,4-diazepan-5-one