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{1-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]cyclopropyl}methanol
methyl 1-cyclohexyl-2-oxo-3-(pyrimidin-5-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
3-{2-[methyl(thian-4-yl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-{5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
2-(cyclopentylmethyl)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-1,6-dimethyl-1,4-dihydropyridin-4-one
N-(furan-3-ylmethyl)-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
6-(2-ethoxypyridin-3-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
8-(4-cyclobutyl-6-methylpyrimidin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(1H-indol-5-yl)-1-methyl-1-(oxolan-3-ylmethyl)urea
3-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]benzonitrile
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(5-{1-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
[5-({4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-(2-aminopyrimidin-5-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,7-dimethylquinoline-4-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
ethyl 4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
5-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}-2-methoxyphenol
(3S,4R)-3-benzyl-4-methyl-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-ol
N-[(2-methoxyphenyl)methyl]-2-(4-oxocyclohexyl)-N-propylacetamide
1-methyl-2-(5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1H-imidazole
N-(1H-indol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-({1-[(4-methylphenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)piperidin-3-ol
(propan-2-yl)({[2-(quinolin-5-yl)phenyl]methyl})amine
(3S,4S)-N-(2,4-dimethoxyphenyl)-3,4-dihydroxypiperidine-1-carboxamide
N-butyl-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(thiophen-3-ylmethyl)acetamide
3-[(cyclohexylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-pyrazol-1-yl)propan-1-one
1-(1H-imidazol-2-ylmethyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
[2-fluoro-5-(pyrimidin-5-yl)phenyl]methanol
2-{1-[(4-fluorophenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-(1H-imidazol-2-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}quinolin-6-yl)acetamide
(3aS,6aS)-2-cyclopentyl-5-(2,4-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
3-{1-[(6-methylhept-5-en-2-yl)amino]ethyl}adamantan-1-ol
N-[(7-{7-methylthieno[3,2-d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amine
2-(2-chlorophenyl)-2-{[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
2-(4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)pyridine
1-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-3-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)urea
(1S,3R)-3-amino-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]cyclopentane-1-carboxamide
(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
N-[(5-methylpyrazin-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
ethyl 1-(1-methoxypropan-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol