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5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
(2R,6S)-4-(5-{1H-imidazo[4,5-b]pyridin-2-yl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-2,6-dimethylmorpholine
N-cyclohexyl-2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]acetamide
4-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]pyridin-3-ol
N-(5-chloro-2-methoxyphenyl)-3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}propanamide
N-[(1R,3R)-3-aminocyclopentyl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
2-cyclopentyl-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-N,N-dimethylacetamide
2-(3-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)acetamide
2-(4-fluorophenyl)-N-{[4-hydroxy-1-(pyridin-3-ylmethyl)azepan-4-yl]methyl}acetamide
5-{3-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-(naphthalen-2-ylmethyl)piperidin-4-ol
N-[2-(2-chlorophenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-4-(pyridin-3-yl)pyrimidine
N-[2-(ethanesulfonyl)ethyl]-3-(4-hydroxyphenyl)benzamide
2-(4-methyl-1H-imidazol-5-yl)-1-[2-(propylsulfanyl)phenyl]-1H-imidazole
5-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
3-[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
4-[5-(3-fluoropyridin-4-yl)furan-2-carbonyl]morpholine
1-[6-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridin-3-yl]ethan-1-one
6-fluoro-2-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
1-(2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
6-[methyl(1-methylpiperidin-4-yl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
(4aS,8aR)-6-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-benzyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
4-[3-(propoxymethyl)pyrrolidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
4-[(2-cyclohexylpyrimidin-5-yl)methyl]morpholine-2-carboxylic acid
7-(5-methylthiophen-2-yl)-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1H-1,3-benzodiazole
1-ethyl-4,6-dimethyl-N-[2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}-6-methylpyridin-3-ol
2-cyclopentyl-1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(dimethylamino)-2-(4-methylphenyl)acetamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzamide
N-cyclopropyl-2,6-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-4-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
1-({4-methyl-5-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-9-(morpholine-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N-methyl-N-phenyl-2-[2-(pyridin-3-yloxy)acetamido]benzamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(3,4-difluorophenyl)-N-methylacetamide
2-cyclopentyl-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
2-[(2-amino-5-butyl-6-methylpyrimidin-4-yl)amino]-1-(pyridin-2-yl)ethan-1-ol
3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-5-phenyl-1,2-oxazole