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(3aS,6aR)-5-(2-aminopyridine-4-carbonyl)-3-[2-(3-chlorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-phenyl-3-(pyridin-2-yl)propanamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
(4S,4aS,8aS)-1-[(2-chloro-6-fluorophenyl)methyl]-4-phenyl-decahydroquinolin-4-ol
[2-(dimethylamino)ethyl](methyl)(2-{[6-(trifluoromethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)amine
ethyl 4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxylate
4-{1-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-imidazol-2-yl}quinoline
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
1-{2-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
N-[(4-chlorophenyl)methyl]-1-[2-(dimethylamino)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(1S,5R)-3-(pyrimidin-2-yl)-6-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2-oxazole-3-carboxamide
N-{2-[2-(4-fluorophenoxy)ethyl]phenyl}cyclopropanecarboxamide
(4aR,8aR)-1-(naphthalene-1-carbonyl)-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridine
2-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(2S)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pentanamide
2-methyl-6-{5-[(2-methyl-1H-imidazol-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}pyridine
1-{4-[(propan-2-yl)amino]pyrimidin-2-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-phenoxypropan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
1-[(3-{[3-(hydroxymethyl)-2-methylphenyl]carbamoyl}phenyl)methyl]-N-methylpyrrolidine-3-carboxamide
4-methyl-N-{2-[7-(5-propyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-4-[4-(methylsulfanyl)benzoyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
[(4-cyclopropyl-5-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(4-chloro-2-methylphenoxy)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}acetamide
2-methyl-9-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(propan-2-yloxy)acetamide
3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
(2R,3S,6R)-5-(1H-imidazol-2-ylmethyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-hydroxy-N-[(6-methylquinolin-5-yl)methyl]pyrazine-2-carboxamide
1-ethyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
9-(2-methyloxane-2-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-{1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carbonyl}piperazin-2-one
4-(4-methoxypyrimidin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethan-1-one
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
(2R,3R,6R)-5-(2-methoxyethyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetamide
4-[(2-hydroxyethyl)sulfanyl]-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
N-ethyl-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
5-[2-(methylsulfanyl)ethyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-[1-(dimethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(5-methyl-4H-1,2,4-triazol-3-yl)-1-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]urea
3-hydroxy-3-({[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(1-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol