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1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-N-cycloheptylpiperidine-4-carboxamide
1-benzyl-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-({4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(trifluoromethyl)morpholine
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
N-[(2R,3R)-1'-[2-(cyclohex-1-en-1-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
2-(dimethylamino)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(3-methylphenyl)acetamide
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(prop-2-en-1-yl)-N-(propan-2-yl)acetamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
1-(2-hydroxyethyl)-N-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
(4aS,7aR)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-cyclopropanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
3-(morpholine-4-sulfonyl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidin-4-amine
2-({2-[(2-hydroxyethyl)[(2E)-3-phenylprop-2-en-1-yl]carbamoyl]phenyl}amino)acetic acid
5-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
5-{1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
N-(4-{[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]methyl}phenyl)acetamide
N2,N2-dimethyl-N5-(propan-2-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-1H-1,3-benzodiazole
(3S,4R)-4-(4-fluorophenyl)-1-(5-methyl-1H-indazole-3-carbonyl)pyrrolidine-3-carboxylic acid
(1-{1-[3-(3-methoxyphenyl)benzoyl]piperidin-4-yl}ethyl)dimethylamine
1-[4-(1,4-diazepan-1-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(2,5-dihydro-1H-pyrrole-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
4-(2-methoxyphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-fluoro-N,N-dimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-methyl-4-[4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenyl]butan-2-ol
N-(4-methoxy-3-pentanamidophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methyl-5-({5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)pyrazine
N-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)acetamide
5-(2-chlorophenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]furan-2-carboxamide
3-(4-chloro-2-methoxy-5-methylphenyl)-1-[(4-fluorophenyl)methyl]-1-(3-hydroxypropyl)urea
1-(azepan-1-yl)-2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]ethan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
5-ethyl-1'-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[4-(benzylamino)piperidin-1-yl]-N-[(2-fluorophenyl)methyl]benzamide
N-[(4-methoxyphenyl)methyl]-1-methyl-N-(pyridin-2-ylmethyl)azepane-2-carboxamide
2-[2-chloro-4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]acetamide
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(2,2-diphenylcyclopropyl)methyl]-1λ6-thiomorpholine-1,1-dione
1-ethyl-N-[(3-methoxyphenyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-(propan-2-yl)piperidine
2-(8-methoxyquinolin-5-yl)phenol
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
3-{[cyclopropyl(ethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione