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3-[5-(1-cyclopropanecarbonylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
2-(6-aminopyridine-3-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
6-fluoro-2-({[1-(1,3-thiazol-5-yl)propan-2-yl]amino}methyl)quinolin-4-ol
1-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(1,2,3-thiadiazol-5-yl)urea
N-[(2-phenoxypyridin-3-yl)methyl]oxane-4-carboxamide
1'-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-ethyl-1,3-thiazole-5-carboxamide
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-{ethyl[(1-ethylpyrrolidin-3-yl)methyl]carbamoyl}-5-methoxybenzoic acid
4-{4-[(carbamoylamino)methyl]-1H-1,2,3-triazol-1-yl}-N-cycloheptylpiperidine-1-carboxamide
4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydrophthalazin-1-one
4-{[1-(cyclohexylmethyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
(3R,4R)-4-(azepan-1-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-ol
[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
2-({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-4-({1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1,3-thiazol-2-amine
1-[(1R,5R)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(cyclopropylmethyl)-N-(2-methoxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrazine
6-(2-fluoro-5-methoxyphenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
(2R,3R,6R)-5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}piperidine-2-carboxamide
1-acetyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
7-chloro-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}quinolin-4-amine
1-{2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
(3S,9aR)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(5-chloropyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
4-hydroxy-N-[2-(methylsulfamoyl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N,N-diethyl-1-[1-(4-{[(2-fluorophenyl)methyl]carbamoyl}phenyl)piperidin-4-yl]piperidine-3-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[5-(4-phenyloxan-4-yl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-N-methylpyridin-2-amine
(1R,7S)-3-(4-fluoro-2-methylphenyl)-6-[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-tert-butyl-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-hydroxypyrimidine-5-carboxamide
N-ethyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
7-(3-chlorophenyl)-4-[(2,2-dimethyloxan-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(4-hydroxypiperidine-1-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-(1H-indol-5-yl)pyridine-4-carboxamide
2-[({1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
7-[3-(1H-indol-3-yl)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-benzyl-3-{1-[2-(morpholin-2-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-ethyl-8-[4-(4-fluorophenyl)-4-oxobutyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,4-dimethylpiperazine-1-carboxamide
7-(cyclobutylmethyl)-2-(1-ethyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide