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2-(1,4-dimethylpiperazin-2-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
methyl 2-[4-(oxan-4-ylmethyl)-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepane-1-carbonyl]benzoate
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-[3-fluoro-5-(propan-2-yloxy)phenyl]pyridin-4-amine
1-{[3-(oxolan-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
5-(azepane-1-carbonyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)benzonitrile
N-{[2-(azepan-1-yl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)furan-3-carboxamide
(3S,9aR)-8-(4-fluorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-5-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
(cyclopropylmethyl)({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
6-(methoxymethyl)-1-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(1R)-1-[3-(2,6-dimethoxyphenyl)phenyl]ethan-1-amine
5-ethyl-N-(3-methoxypropyl)-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-chloro-6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
N-(2,5-dimethylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)propanamide
3-(2-ethylpiperidine-1-carbonyl)-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-1,4-dihydropyridin-4-one
1-{[5-(1-cyclopentylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
6-methoxy-N-(2-methoxyethyl)-3-methyl-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
1'-{[(1s,4s)-4-aminocyclohexyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-cyclopropyl-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-(naphthalen-2-yloxy)-1-[(propan-2-yl)carbamoyl]piperidine-4-carboxylic acid
2-methyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-N-(2-hydroxyethyl)-2-(4-methylphenyl)-N-propylacetamide
9-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methyl-3,9-diazaspiro[5.6]dodecane
4-(1,3-dihydroxypropan-2-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(1H-pyrazole-4-sulfonyl)piperidin-3-yl]propanamide
(4aS,7aR)-1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-[(cyclopropylmethyl)(methyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
1-(4-aminopyrimidin-2-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-[1-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
1-{1-[2-(3-methylphenyl)benzoyl]piperidin-4-yl}piperidin-4-ol
9-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-ethyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
(3S)-3-benzyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-(oxan-4-yl)-3-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
N-[2-(azepane-1-carbonyl)phenyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
5-{[methyl({[3-(2-{4-[3-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
3-[1-(2,1,3-benzoxadiazole-4-sulfonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,9aR)-8-(3,5-difluorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl (2S,4R)-1-(1-benzylpiperidin-4-yl)-4-(2-cyclopropylquinoline-4-amido)pyrrolidine-2-carboxylate