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1-(5-ethyl-1H-pyrrole-2-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(cyclopropylmethyl)-N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(4-ethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-(pyridin-2-yl)-5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
N-[(3S,5S)-1-(2-ethoxyacetyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethylpyrimidine-5-carboxamide
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-(4-methoxyphenyl)-1H-pyrazole
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
(2-methoxyethyl)(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)(pyridin-2-ylmethyl)amine
1-benzyl-4-ethyl-1,4-diazepan-5-one
N'-cyclohexyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N'-methylbutanediamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
2-ethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
3,5-dimethyl-1-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
3-[(2-hydroxyethyl)({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amino]-3-methyl-1λ6-thiolane-1,1-dione
5-chloro-2-fluoro-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}benzamide
N-[2-(dimethylamino)ethyl]-N-ethyl-7-fluoro-2-methylquinoline-4-carboxamide
4-{2-methyl-6-[1-(4-methylpent-3-en-1-yl)piperidin-3-yl]pyrimidin-4-yl}morpholine
[1-({1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(pyridin-4-ylmethyl)pyridin-2-amine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]propanamide
1-methyl-3-phenyl-5-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1H-pyrazole
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
2-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}benzene-1,3-diol
3-[(2-methoxyethyl)sulfamoyl]-5-(quinolin-6-yl)benzoic acid
3-{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
[(2-methoxyphenyl)methyl](prop-2-en-1-yl){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
3-cyclopropyl-1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(3-methylthiophen-2-yl)methyl]urea
6-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(1-benzofuran-2-yl)-1-methyl-1H-pyrazol-5-amine
(3aS,6aS)-2-[(3-fluorophenyl)methyl]-5-(oxane-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-hydroxypropyl)-1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-1-phenylcyclohexane-1-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-3-(pyrrolidine-1-carbonyl)-1H-pyrazole
1-{2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}ethan-1-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}piperidine-3-carbonitrile
2-{2-[2-(3-fluorophenyl)azepan-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
ethyl 1-[(4-methoxyphenyl)methyl]-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-chloro-4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)oxan-4-amine
(1R,5R)-N,N-dimethyl-6-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[2-(methylamino)ethyl]pyrimidin-2-amine
3-benzyl-7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
methyl (2S,4R)-4-acetamido-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidine-2-carboxylate
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-(1-cyclohexyl-3-phenyl-1H-1,2,4-triazol-5-yl)-1-(2-methoxyethyl)pyrrolidin-2-one
4-phenyl-1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-4-ol