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N-[(5-oxopyrrolidin-2-yl)methyl]-2-(3-phenylpropyl)-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-ethyl-3-methyl-8-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(adamantan-1-yl)-1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(1-methyl-1H-pyrazol-4-yl)-1-[2-(1-methylpiperidin-2-yl)ethyl]-1,2,3,6-tetrahydropyridine
3-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-{[4-(hydroxymethyl)phenyl]methyl}-3-(1H-imidazol-2-yl)benzamide
2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(thiophen-2-ylmethyl)acetamide
(3S,4S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-methylpiperidine-3,4-diol
[(3R,4R)-1-(2-fluoro-4-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
ethyl 3,5-dimethyl-4-({1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)-1H-pyrrole-2-carboxylate
3-chloro-N-cyclopentyl-4-{[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
4-{2-[(2-methoxyethyl)carbamoyl]ethyl}-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(pyridin-3-yloxy)ethan-1-one
methyl (2S,4R)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(dimethylamino)pyrrolidine-2-carboxylate
4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
6-cyclopentyl-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-2-amine
3-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-1-[(3-methylphenyl)methyl]urea
3-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-ylmethyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-(2-methoxyethyl)-2,8-diazaspiro[4.5]decan-3-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
N-benzyl-N-methyl-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
ethyl 4-[(4-{[1-(3-chloro-4-fluorobenzenesulfonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
7-(2-chlorobenzenesulfonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
(1S,5R)-3-benzyl-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(6-methylpyridin-2-yl)methyl]amine
4-{1-methyl-3-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-5-yl}morpholine
6-fluoro-3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinolin-4-ol
3-ethyl-1-[2-(thiophene-2-sulfonamido)acetyl]piperidine-3-carboxylic acid
4-({1-[3-(1-methylpiperidin-3-yl)propanoyl]azetidin-3-yl}oxy)benzoic acid
3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)benzoic acid
methyl (2S,4S)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
N-cyclopropyl-1-{2-[(2-methylphenyl)sulfanyl]acetyl}piperazine-2-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-phenylpiperazine
N-(3,5-dimethylphenyl)-6-[2-(1H-imidazol-1-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]acetamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
(3aS,6aR)-5-(5-chloropyridin-2-yl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclopentanamine
4-(3-benzyl-1H-pyrazol-5-yl)-1-(furan-2-carbonyl)piperidine
1-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-(quinolin-2-ylmethyl)acetamide