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3-{2-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-{4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]piperidin-1-yl}ethan-1-one
3-methyl-N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
2-(1-ethylpiperidin-4-yl)-N-(1-phenylpiperidin-4-yl)acetamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(9H-purin-6-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(ethylsulfanyl)ethyl]-6-{methyl[(2-methylphenyl)methyl]amino}-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
N-methyl-2-(pyridin-2-yl)-N-(pyrimidin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperazin-1-yl)quinazoline
(1s,4s)-4-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
2-butyl-N-[(3-fluorophenyl)methyl]-4-methyl-3-oxopiperazine-1-carboxamide
N-(adamantan-2-yl)-6-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1,4-dimethyl-9-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecane
5-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxybenzoic acid
3-({[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
(3R,4R)-1-cyclohexyl-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-[2-(2-fluorophenyl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
(1S,5R)-6-benzyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrrolidine-1-sulfonamide
3-methyl-7-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
(3S,4R)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-methylpiperidine-3,4-diol
3-{5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
N-[2-(1H-indol-3-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-butyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
5-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
4-{5-[2-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)ethyl]-1-propyl-1H-1,2,4-triazol-3-yl}benzamide
1-(2-phenylbenzoyl)azepan-4-amine
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(prop-2-ene-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]ethyl}morpholine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(2,5-dimethylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-fluoro-N,1,3-trimethyl-1H-indole-2-carboxamide
1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(piperidine-1-carbonyl)piperidine
3-(3-{3-[5-(trifluoromethyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
2-[1-cyclopentyl-4-(3-cyclopentylpropyl)piperazin-2-yl]ethan-1-ol
2-(2-chloro-4-fluorophenoxymethyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-methyl-2-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,2-dihydroquinoline-4-carboxamide
(3S,4R)-3-cyclopropyl-N,N-dimethyl-4-[3-(1H-pyrazol-1-yl)benzamido]pyrrolidine-1-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(1-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrazine-2-carboxamide
1-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}benzonitrile
(4aS,8aR)-6-(6-oxo-1,6-dihydropyridine-3-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(5-methanesulfonamido-2-methylphenyl)-3-(2,2,2-trifluoroethyl)urea
5-chloro-6-[3-(1-methoxyethyl)phenyl]pyridine-3-carboxylic acid