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2-(azepan-1-yl)-N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-oxoacetamide
1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
N-(3-cyclopentylpropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-(pyrimidin-2-yloxy)benzamide
dimethyl[3-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)propyl]amine
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
N-(1-{1-[(6-chloropyridin-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)furan-2-carboxamide
6-methyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
ethyl 1-[(3-chloro-4-hydroxyphenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
(3R,4S)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-propylpyrrolidin-3-amine
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,6-dimethylpyrimidin-2-amine
4-methyl-2-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,3-thiazole-5-carboxamide
N-[2-(dimethylamino)-3-methylbutyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
{2-[2-(hydroxymethyl)phenyl]-8-methylquinolin-3-yl}methanol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(1,3-benzothiazol-2-yl)piperidin-3-amine
6-{[4-(2-phenylazetidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-(1H-indol-2-ylmethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{[5-(oxolan-2-yl)thiophen-2-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
1-[(4-methylphenyl)methyl]-5-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-3-carboxamide
2-chloro-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-(trifluoromethyl)benzamide
4-(1H-pyrazol-1-yl)-6-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
3-(1-ethyl-1H-imidazol-2-yl)-1-(4-methanesulfonylbenzoyl)piperidine
(3R,4R)-4-amino-1-(3-aminothiophene-2-carbonyl)piperidin-3-ol
1-(4-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[2-(oxolan-3-yl)ethyl]benzamide
2-fluoro-N-[3-hydroxy-1-(4-methylphenyl)propyl]-5-sulfamoylbenzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]propan-1-ol
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
2-(3-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
7-(5-chloropyridin-2-yl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(7-fluoro-2-methylquinoline-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-cyclopentanecarbonyl-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(1-methyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
(1S,5R)-6-(benzenesulfonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(1,3-benzothiazol-2-ylmethyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-methoxy-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-{2-oxo-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}azepan-2-one
3-benzyl-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-(2-ethoxyphenyl)-1-(1-methylpiperidin-4-yl)-1-(pyridin-4-ylmethyl)urea
7-methoxy-3-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
3-(2-{methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1,3-dimethyl-7-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]ethyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
1-[(4-chlorophenyl)methyl]-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-cycloheptylpropanamide