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N-methyl-1-(pyrazine-2-carbonyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
N-[2-(2-chlorophenoxy)ethyl]-N'-(4-methylphenyl)propanediamide
2-{[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]amino}-1-(3,4-dimethoxyphenyl)ethan-1-ol
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(2-phenylethyl)piperidin-1-yl]propan-1-one
N4,N4,5-trimethyl-N2-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrimidine-2,4-diamine
2-(4-fluorophenoxymethyl)-N-(3-hydroxy-3-methylbutyl)-N-methyl-1,3-oxazole-4-carboxamide
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(carbamoylmethyl)pyrrolidine-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(6-methoxynaphthalene-2-carbonyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine
N-[(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
1-(furan-2-yl)-2-[2-(3-phenylpropyl)morpholin-4-yl]ethane-1,2-dione
N-[2-(1H-indol-3-yl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-{4-[6-(dimethylamino)pyridazin-3-yl]phenyl}propanoic acid
1-(3,5-dimethylphenyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-2-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
5-(3-fluorophenoxymethyl)-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
N-methyl-3-(morpholine-4-carbonyl)-1-propyl-N-(1,3-thiazol-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)pyrrolidin-2-one
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
7-methyl-2-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-6-[4-(1H-pyrazol-5-yl)phenyl]pyridine-3-carboxamide
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-(pyridin-3-yloxy)ethan-1-one
(3S)-3-({[3-methoxy-5-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}amino)azepan-2-one
(3S,4S)-1-(3-ethyl-1H-indole-2-carbonyl)-4-methylpiperidine-3,4-diol
N-[2-(1H-imidazol-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-1'-[2-(methylamino)pyridine-3-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]phenyl}prop-2-yn-1-ol
N-[4-(5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenyl]acetamide
2-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}propan-2-ol
N-[3-(4-butyl-3-oxopiperazin-1-yl)-3-oxopropyl]-4-fluorobenzamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[3-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
1-(2,3-dimethylphenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-amine
4-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]benzene-1-sulfonamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
3-phenyl-5-[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
2-(3-chlorophenyl)-2-hydroxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-methoxy-N-(pyridin-3-ylmethyl)propanamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine
methyl (2S,4R)-1-(3-chloropyridine-4-carbonyl)-4-(dimethylamino)pyrrolidine-2-carboxylate
5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazole
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
2-{[(3-ethoxyphenyl)methyl](4,4,4-trifluorobutyl)amino}ethan-1-ol
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(2S)-1-[4-(3-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[1-(6-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxylate
N-(3,5-dimethylphenyl)-4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
N-ethyl-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide