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N,N-diethyl-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
{2-[4-(3-ethynylbenzoyl)morpholin-2-yl]ethyl}dimethylamine
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-(2,2-diphenylethyl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
N-{2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]thiophen-3-yl}acetamide
3-{5-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
7-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2-methylphenyl)methyl]piperidin-3-ol
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
1-propyl-4-{[2-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}piperidine
[9-(3-methoxypropyl)-3-(1H-pyrrole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
3-(2,4-difluorophenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
4-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-cyclopentyl-1,3-dimethyl-N-propyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3-methylpyridin-4-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
4-(4-cyclopentylpyrimidin-2-yl)phenol
4-[(1-ethyl-1H-indol-6-yl)methyl]-1-methylpiperazine-2-carboxylic acid
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-5-methylpyrazine-2-carboxamide
1-(1-benzofuran-3-carbonyl)azocane
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
N-[(3S,4R)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-{benzyl[(1-methylcyclopropyl)methyl]amino}propan-1-ol
N-cyclopentyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]thiophen-3-yl}acetamide
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-7-fluoro-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
9-[(2-ethylpyrimidin-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]piperidin-4-yl}-N-methylacetamide
6-[(diethylamino)methyl]-N-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 4-({[(3S,5S)-1-benzyl-5-(methylcarbamoyl)pyrrolidin-3-yl]amino}methyl)benzoate
1-(1H-imidazol-4-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4,6-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
4-(1H-imidazol-1-ylmethyl)-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine
N-[(2R,3R)-1'-[(2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-cyclopentyl-3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
1-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
4-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-(dimethylamino)-2-(2-methylphenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
2-(dimethylamino)-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-2-(4-methylphenyl)ethan-1-one
4-({5-[1-(cyclopropylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(2-chlorophenyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-2-hydroxyacetamide