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4-{1-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]ethyl}morpholine
1-{3-[(pyrimidin-2-yl)amino]propyl}piperidin-4-ol
N-(1-methanesulfonylpiperidin-4-yl)-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-methyl-5-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(2-phenylethyl)morpholine
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
(1S,6R)-9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
7-methyl-2-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-cyclobutyl-2-(dimethylamino)-2-(2-methylphenyl)acetamide
N-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[1-benzyl-4-(propan-2-yl)piperazin-2-yl]ethan-1-ol
1-(2,3-difluoro-6-methoxybenzoyl)-4-(2-methylphenyl)-1,4-diazepane
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
1-methyl-2-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,8-naphthyridine-2-carboxamide
methyl (1S,3S,3aR,6aS)-3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-(2,6-difluoro-3-methylbenzoyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-(methoxymethyl)-N,1-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-({1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
4-[(4-methylphenyl)methyl]-11-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)benzamide
1-{6-[4-(3-methoxybenzoyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
N-methyl-5-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)furan-2-carboxamide
4-(benzyloxy)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]butanamide
N-[(3S,5S)-1-methyl-5-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidin-3-yl]morpholine-4-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidine-2-carboxamide
N-(diphenylmethyl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(4-chlorophenyl)butan-1-one
N-{3-methyl-4-[2-(trifluoromethyl)morpholine-4-carbonyl]phenyl}acetamide
(4S)-3,3,4-trimethyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-ol
N-{[1-(dimethylamino)cyclohexyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
methyl 8-{[4-(benzyloxy)phenyl]methyl}-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[cyclopentyl(methyl)amino]ethan-1-one
3-[(dimethylamino)methyl]-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-ol
2-{4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}pyridine
2-{4-[(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrazine
2-ethyl-2-{[methyl({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}butan-1-ol
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[4-(pyridin-3-yloxy)phenyl]urea
methyl 7-oxo-9-(propan-2-yloxy)-3-(thiolan-3-yl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazole
3-(2-amino-1,3-thiazol-4-yl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}propan-1-one
3-(oxolan-3-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
N,N,7-trimethyl-3-{[(2-phenylethyl)amino]methyl}quinolin-2-amine