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1-[(5-ethylpyridin-2-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
dimethyl(3-{2-[1-(4-methylpyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-benzyl-N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
1-(4-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}phenyl)-1H-1,2,3,4-tetrazole
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-phenylacetamide
4-{5-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,5-dimethyl-1H-pyrazole
N-cyclopentyl-4-(1H-pyrazol-1-yl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)benzamide
2-(2,5-dimethylphenoxy)-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]propanamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-{[(2S,4S)-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide
5-(quinolin-8-yl)thiophene-2-sulfonamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
6-chloro-2-{[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-1,3-benzodiazole
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-fluoroquinolin-3-yl}methyl)[2-(1H-imidazol-1-yl)ethyl]amine
2-tert-butyl-7,7-dimethyl-N-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-5,6,7,8-tetrahydroquinazolin-5-amine
3-benzoyl-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
[(2S,6S)-4-(2,3-dimethyl-1H-indole-7-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(1s,4s)-4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-amido]cyclohexane-1-carboxylic acid
3-[(3R,4S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperazine-2-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})methylamine
N-ethyl-6-(4-fluorophenyl)-N-[2-(pyrrolidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-ethyl-6-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-hydroxy-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}ethan-1-one
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-3-methylimidazolidin-2-one
2-methyl-4-{4-[3-(pyrrolidin-1-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
3-(3-chloro-4-propoxyphenyl)-1-(1,4-dioxan-2-ylmethyl)-1-methylurea
(2H-1,3-benzodioxol-5-ylmethyl)[(2E)-3-(furan-2-yl)prop-2-en-1-yl](pyridin-3-ylmethyl)amine
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-amine
3-({[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-(pyridin-3-yloxy)acetamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-methyl-4-phenyl-3-(1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2,6-dimethoxypyridine-3-carboxamide
3-(4-fluorophenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
2-methyl-3-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[2-(pyridin-2-yl)piperidin-1-yl]butan-1-one
methyl (2R,4S)-1-cyclohexanecarbonyl-4-hydroxypiperidine-2-carboxylate
N-(3-{4-[(2,2-diphenylethyl)amino]piperidin-1-yl}phenyl)pyridine-4-carboxamide
2-(carbamoylamino)-N-[(3R,4S)-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
[2-(5-aminopyridin-3-yl)-7-methylquinolin-3-yl]methanol
7-(cyclopropylmethyl)-2-(5-ethylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,4-dimethoxyphenyl)-3-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-indole
methyl (2S,4S)-4-cyclohexaneamido-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate