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(3aS,6aS)-5-(1-benzofuran-5-ylmethyl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1S,5R)-6-(4-chloro-2-methylbenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-amino-N,N-diethyl-1-[(2R)-2-hydroxy-3-methylbutanoyl]pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
N-[(2-chlorophenyl)methyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpyrimidine-5-carboxamide
2-[(furan-2-ylmethyl)({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]butan-1-ol
7-fluoro-N,N-dimethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(3aS,6aS)-2-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(4-fluorophenyl)methyl]-4-hydroxy-N-(2-hydroxyethyl)-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-amino-1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(methylsulfanyl)ethan-1-one
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}benzenesulfonyl)piperidine
3-(1-cyclopentanecarbonylpiperidin-3-yl)-N-(4-fluoro-2-methylphenyl)propanamide
2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N,N-dimethyl-2-{[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
8-cyclobutanecarbonyl-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
8-[(3-chlorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclohex-1-ene-1-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
1,3-dimethyl-2,6-dioxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{4-[2-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}propan-1-one
6-{3,9-diazaspiro[5.6]dodecan-9-yl}-N-ethylpyridine-3-carboxamide
3-amino-1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidine-3-carboxylic acid
(propan-2-yl)({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-phenylacetamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(pyrazin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2,6-dimethyl-4-({[2-(pyridin-3-ylformamido)ethyl]amino}methyl)phenyl acetate
[(2S,6S)-4-(3-fluoropyridin-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
6-(8-methylquinolin-5-yl)pyridin-3-ol
2-(oxolan-2-ylmethyl)-9-(pyridazine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{[1-(3-methylbutyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperazin-1-yl)ethan-1-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
2-(methylsulfanyl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperazine-1-sulfonamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(pyridin-2-ylsulfanyl)acetamide
2-methyl-N-(2-{[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}phenyl)furan-3-carboxamide
1-cyclopentyl-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-5-phenylpentan-1-one
4-hydroxy-N-(4-methanesulfonylphenyl)-4-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
methyl 5-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-cyclopropyl-1-[1-(cyclopropylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-(2-oxoazepan-3-yl)propanamide