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2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1,3-benzoxazole
1-(5-{[2-(methoxymethyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-4-methyl-1,4-diazepane
N-[2-(4-fluorophenyl)-1-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine
5-chloro-2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
(1-{[4-(difluoromethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-methyl-7-(methylsulfanyl)-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
N-[(2-methoxyphenyl)methyl]-2-[2-(2-methylphenyl)pyrrolidin-1-yl]acetamide
7-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
7-methoxy-2-(1H-pyrazol-4-yl)-4-(thiomorpholine-4-carbonyl)quinoline
3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
7-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-4-methyl-2H-chromen-2-one
N-(3,4-dimethylphenyl)-1-(4-methoxybenzoyl)piperidin-3-amine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methylacetamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-3-phenyl-1,2-oxazole
N-[3-(4-{[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
3-methoxy-1-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,2-dihydropyridin-2-one
2-{[2-(4-chlorophenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-ethoxy-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
3-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(4-fluorophenyl)methyl]propanamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)benzamide
2-{5-[2-(3,4-dimethyl-1H-pyrazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
2-methoxy-N-({3-methyl-7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
6-(2-chlorophenyl)-N-[(2S)-2,3-dihydroxypropyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl({[4-(methylsulfanyl)phenyl]methyl})(oxan-2-ylmethyl)amine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(1S,5R)-6-(3-chloro-4-methylbenzoyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}[(2-methylphenyl)methyl](prop-2-en-1-yl)amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[3-(2-methoxyacetamido)phenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-3-(hydroxymethyl)phenyl}methanol
ethyl[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
4-ethyl-3-(piperidin-3-yl)-1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N-(2-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}ethyl)pyridin-4-amine
N-({3-[3-methyl-7-(thiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyrrolidine-1-carbonyl)piperidin-3-yl]methanol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-[2-(2-chlorophenyl)-1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[(1-cyclooctylpyrrolidin-3-yl)methyl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
2-(1H-indol-1-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-[3-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[1-(2-phenylethyl)-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl]ethan-1-ol