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3-[(1-ethyl-5-oxopyrrolidin-3-yl)sulfamoyl]-N-(2-methoxyethyl)-N-methylbenzamide
N-[2-({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}amino)ethyl]-4-methylpyridin-2-amine
N-[2-(4-methoxyphenyl)ethyl]-1,2,5-trimethyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-3-carboxamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
methyl 3-({[1-(4-chlorophenyl)cyclobutyl]formamido}methyl)-5-(furan-2-amido)benzoate
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
2-butyl-8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-methoxy-4-{1-oxa-8-azaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
2-[2-methyl-3-({[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
3-(2-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}ethyl)pyridine
N-ethyl-2-(1-ethyl-3-oxopiperazin-2-yl)-N-[2-(4-fluorophenoxy)ethyl]acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
[(1-cyclopentylpiperidin-4-yl)methyl][(5-ethylfuran-2-yl)methyl](pyridin-3-ylmethyl)amine
6-{3-oxo-3-[4-(quinazolin-4-yl)piperazin-1-yl]propyl}-2,3-dihydropyridazin-3-one
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzenesulfonamide
(3S,4R)-N,N-dimethyl-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
N-benzyl-3-{[(1,4-dioxan-2-ylmethyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(oxolane-2-carbonyl)piperazine
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl[4-(morpholin-4-yl)butyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,7,8-trimethylquinoline-4-carboxamide
2-{4-cyclopentyl-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{4-[(1-ethyl-1H-indol-3-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-({[(3R,4R)-1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-methylpiperidin-3-amine
1-[(2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-[(3,4-dimethoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-{4-[(3R)-3-hydroxypyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)ethan-1-one
2-{5-[6-(piperidin-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(pyridin-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(diethylamino)-3-(2-methoxy-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-acetyl-8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-(2-chloro-6-fluoro-3-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridazin-3-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(phenylsulfanyl)ethan-1-one
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-4-[(2-hydroxyethyl)sulfanyl]benzamide
3-(4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
4-(6-methoxypyridin-2-yl)-2-({[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]amino}methyl)phenol
4-(2-methylphenoxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
2-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl)acetic acid
(4aS,8aR)-6-[3-(1H-imidazol-2-yl)benzoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid