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1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-ol
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-N'-(3-ethylphenyl)butanediamide
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-3-carboxamide
N-(3-methoxypropyl)-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(3S,5S)-1-[2-(dimethylamino)acetyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrazine-2-carboxamide
N-methyl-5-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-ethyl-7-(2-methoxybenzamido)-1-methyl-N-[3-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-5-carboxamide
2,3-dimethyl-N-(6-methylpyridin-3-yl)quinoxaline-6-carboxamide
1-tert-butyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]piperidine-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,4R)-4-methyl-3-(propan-2-yl)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]pyrrolidin-3-ol
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
4-(4-methoxy-2-methylphenyl)-5-(propan-2-yl)pyrimidine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
2-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-4-amine
1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
3-{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
2-{5-[2-(morpholin-4-yl)pyrimidin-5-yl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(2-methylpropyl)-8-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
(3S,4S)-1-(6-methylpyridine-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-oxo-1,2-dihydroquinoline-3-carboxamide
3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[4-(2-cyanophenyl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-(4-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-(trifluoromethyl)pyridin-2-amine
N-(2-methoxyethyl)-6-[4-(2-phenoxyethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(furan-3-ylmethyl)urea
1-(3,3-dimethylcyclohexyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-({6-[(E)-2-phenylethenyl]pyridazin-3-yl}amino)ethan-1-ol
4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)benzoic acid
2-amino-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(diethylamino)ethyl]-1-{2-[(3,4-dimethoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
4-(hydroxymethyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-ol
2-{[(1-benzylpiperidin-4-yl)methyl](methyl)amino}pyridine-4-carboxamide
N-methyl-4-{2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}benzene-1-sulfonamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(morpholin-4-yl)propan-1-one
1-(2-methoxyethyl)-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperazine
6-fluoro-2-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)quinolin-4-ol
4-{5-[1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
5-[2-(furan-3-yl)-1H-imidazol-1-yl]-8-methylquinoline
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(piperidine-1-sulfonyl)benzamide
(3S,4R)-1-[(3-fluoropyridin-4-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol