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3-({[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-[(2-chloro-6-fluorophenyl)methyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-cyclopropanecarbonyl-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{furo[3,2-c]pyridin-4-yl}-4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazine
2-(2-{[2-(2-methoxyphenyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-(2-phenylethyl)-1-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-(2,3-dihydroxypropyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
8-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[6-(pyrimidin-5-yl)pyridazin-3-yl]azepane
2-propyl-N-[1-(thiophen-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
9-[(4-chloro-3-fluorophenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]pyrimidine
N-benzyl-N-methyl-3-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-N'-[2-(propan-2-yl)phenyl]butanediamide
3-[(2R,3R,6R)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-[2-cyclopropyl-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]pyrazine
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-[3-(2,6-dimethylphenoxy)propyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
propyl 2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetate
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(piperidin-1-yl)acetamide
4-chloro-1-ethyl-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
4-(3-fluoropyridin-2-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
2-(adamantan-1-yl)-6-(1-methylpiperidin-4-yl)-3,4-dihydropyrimidin-4-one
(3aS,6aS)-2-[3-(methylsulfanyl)propyl]-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-methylbutyl)-8-(4-methylpiperazine-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
2-(benzyloxy)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
methyl 4-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoate
5-{1-[1-(pyrimidin-2-yl)piperidine-4-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(1-methylpiperidin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-{[7-methyl-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]methyl}-1H-imidazole
N,N-diethyl-1-{2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carbonyl}piperidine-3-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
N-[1-(furan-2-carbonyl)piperidin-3-yl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
(1S,6R)-9-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-methoxypropyl)benzamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridine-3-carboxamide
[(3R,4R)-1-(3-phenylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3R)-N-[(2-fluorophenyl)methyl]-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carboxamide
5-cyclobutyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1,3,4-oxadiazol-2-amine
(2S,4S)-4-cyclohexaneamido-N-ethyl-1-methyl-N-(2-methylprop-2-en-1-yl)pyrrolidine-2-carboxamide
N-(2-cyclopropylphenyl)-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carboxamide