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methyl 3-(cyclobutylmethoxy)-5-{[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)carbamoyl}benzoate
1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-2-methyl-1,4-diazepan-5-one
methyl 3-[(2E)-3-phenylprop-2-enamido]-5-[(pyridin-4-ylformamido)methyl]benzoate
N-tert-butyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3-cyclopropyl-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1H-1,2,4-triazol-1-yl)acetic acid
[2-(4-chlorophenyl)ethyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-[1-(methoxymethyl)cyclobutanecarbonyl]-2-(2-methylphenyl)pyrrolidine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-(furan-2-ylmethyl)-4-{[2-hydroxy-2-(3-hydroxyphenyl)ethyl]amino}pyridine-2-carboxamide
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}furan-2-carboxamide
4-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]thiomorpholine
7-methyl-2-[2-(quinazolin-4-yloxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-acetyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-3-carboxamide
2-amino-1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpropan-1-one
N-ethyl-5-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}pyrimidin-2-amine
1-cyclopentyl-N-[2-(1H-imidazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1'-(2-methoxy-4-methylbenzoyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N,N-dimethyl-1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]azepan-4-amine
6-methyl-4-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
2-[2-(adamantan-1-yl)acetamido]-3-hydroxypropanoic acid
3-(4-chlorophenyl)-5-[(2-cyclopropyl-1H-imidazol-1-yl)methyl]-1,2-oxazole
N-[4-(furan-2-yl)phenyl]-1-[3-(pyridin-2-yl)propanoyl]piperidine-3-carboxamide
N-ethyl-4-(1H-pyrrol-1-yl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
methyl 4-{[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
(3R,5S)-5-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-3-ol
2-(1H-indol-3-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(1H-1,2,3-benzotriazol-5-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-2-yl)ethyl]acetamide
4-cyclobutaneamido-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylbenzamide
methyl[(4-methyl-1,3-thiazol-2-yl)methyl][(1-propyl-1H-imidazol-2-yl)methyl]amine
N-cycloheptyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(4aS,8aR)-6-(2,3-dihydro-1H-inden-2-yl)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-1-yl]acetamide
2-(morpholin-4-ylmethyl)-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,4-oxazepane
(1R,3S)-7-(5-chloro-2-methylpyrimidine-4-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
3-cyclohexyl-1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazole
2-[3-(piperazin-1-yl)phenyl]pyridine-3-carboxamide
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1,3-thiazole-4-carboxamide
1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-(methylsulfanyl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
ethyl 1-(1,4-dithiepan-6-yl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(4aS,8aR)-6-(2-methylpyrimidine-5-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
2-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one