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N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
(1S,5R)-3-cyclobutanecarbonyl-6-(2,6-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-phenylcyclohexane-1-carboxamide
2-(ethoxymethyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(dicyclopropylmethyl)amine
4-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-N-methylpyridin-2-amine
N-[(2,3-dimethoxyphenyl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-methyl-N-(pyridin-3-ylmethyl)aniline
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[(3-methylthiophen-2-yl)methyl]amine
N-{2-[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
(2R,4S)-4-hydroxy-1-(3-methylpyridine-2-carbonyl)piperidine-2-carboxylic acid
N4-ethyl-N2-(morpholin-2-ylmethyl)pyrimidine-2,4-diamine
2-(3-hydroxyphenyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
(2R,3R)-3-[4-(pyrrolidin-1-yl)piperidin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-6-methylpyridin-3-ol
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
3-ethyl-5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-4-carboxamide
7-(2-oxopyrrolidin-1-yl)-4-[2-(prop-2-yn-1-yloxy)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[3-(3-fluorophenyl)phenyl]-1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidine-4-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-ethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2S,4R)-4-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-methylpyrrolidin-2-yl]methanol
1-ethyl-3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(oxan-2-ylmethyl)piperidin-4-amine
6-(2-chlorophenyl)-N-ethyl-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1R,2R,6S,7S)-4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-azatricyclo[5.2.1.02,6]decane
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-cyclopentyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(4aS,7aR)-1-(3-hydroxypropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{2-methyl-7-[(4-methyl-1H-imidazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-oxazepane
2-methyl-N-(4-{[(2S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]oxolan-2-yl]methyl}phenyl)propanamide
1-[6-hydroxy-4-(1H-indol-5-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-5-{1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-butyl-5-cyclopropyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1,3-oxazole-4-carboxamide
N-methyl-4-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-(furan-2-ylmethyl)-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
3-(4-benzylpiperazine-1-carbonyl)-1-(cyclohexylmethyl)-2-(methoxymethyl)-6-methyl-1,4-dihydropyridin-4-one
7-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-2,3,4,9-tetrahydro-1H-carbazol-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,3-difluorobenzamide
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
2-cyclopropyl-8-[(3,5-dimethoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{[(2-chloro-5-methylphenyl)carbamoyl]amino}cyclopentane-1-carboxamide
8-(2,5-dimethylfuran-3-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
[(3R,4R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(1-benzothiophene-5-carbonyl)-2-(1-methyl-1H-pyrazol-3-yl)piperidine
1-(3-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-{3-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole