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1-(furan-2-ylmethyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
3-{2-[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
(2S)-4-methyl-2-phenyl-1-[3-(1H-pyrazol-4-yl)propyl]piperazine
1-(3-methylbut-2-en-1-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-{2-azaspiro[4.4]nonane-2-carbonyl}-N-(oxolan-3-yl)benzene-1-sulfonamide
1-[(4aR,8aR)-4a-hydroxy-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
4-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}morpholine
N-[1-(hydroxymethyl)cyclohexyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
8-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1,3-benzothiazol-2-ylmethyl)-2-cyclopropyl-N-methyl-1,3-benzoxazole-6-carboxamide
2-(1-{[1-(4-chloro-2-methylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-methyl-1,3-benzothiazole-5-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-methyl-5-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
N,N-dimethyl-3-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrazin-2-amine
1-benzyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-[(4-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
(1R,3S,5S)-8-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(6-methyl-2H-1,3-benzodioxol-5-yl)urea
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-cyclopropaneamido-4-methyl-N-{1-[(3-methylphenyl)methyl]cyclopropyl}benzamide
1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-chloro-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyridine-4-carboxamide
N-({1-[(3-ethoxyphenyl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}-2,3,6-trimethylquinoline-4-carboxamide
methyl 3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}benzoate
methyl({[2-(methylsulfanyl)phenyl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
1-(1-benzyl-4-phenylpiperidine-4-carbonyl)azetidine-2-carboxylic acid
2-(pyridin-4-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
N-(carbamoylmethyl)-3-(2-methylphenyl)-3-phenylpropanamide
ethyl 4-({1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)piperidine-1-carboxylate
(3S,4S)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-propylpyrrolidine-3-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
(3aS,6aS)-2-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-cyclohexyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)acetamide
9-methyl-3-(3-methyl-1H-pyrazole-5-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
4-(naphthalen-1-ylmethyl)-1,4-oxazepan-5-one
N-[(2-fluorophenyl)methyl]-3-[1-(3-methoxypropanoyl)piperidin-3-yl]propanamide
N-[(3-methoxyphenyl)methyl]-3-[1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-ol
5-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
2-(dimethyl-1,3-thiazol-5-yl)-N-{2-[(4-fluorophenyl)formamido]ethyl}acetamide
4-[(2-methoxypyridin-3-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-phenylpiperidin-4-ol
{4-[(5-chlorofuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
4-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}pyrimidine