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(4aS,8aS)-2-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-decahydro-2,7-naphthyridine-2-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N4-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(morpholin-4-yl)piperidine-1-carboxamide
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
2-(1H-imidazole-5-carbonyl)-6-methyl-5-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(1H-indazol-5-yl)piperazin-2-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2,7,8-trimethylquinoline-4-carboxamide
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-(2-methoxyphenyl)-2-methylpiperazine
[(2S)-1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidin-2-yl]methanol
5-[5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-[(3-chloro-2-fluorophenyl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
ethyl 2-({5-[(4-methanesulfonamidopiperidin-1-yl)methyl]pyrimidin-2-yl}(methyl)amino)acetate
(4aS,8aR)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)pyrazolo[1,5-a]pyridine-3-carboxamide
(5S,9aS,9bS)-2-(pyridin-3-ylmethyl)-5-[4-(pyrimidin-2-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
(1S,5R)-3-(6-aminopyrimidin-4-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-3-ethyl-4-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
5-(4-fluorophenyl)-N-[2-(piperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
N-[(1-benzylpiperidin-4-yl)methyl]-1-(difluoromethyl)-N-methyl-1H-pyrazole-5-carboxamide
N-{[4-(isoquinolin-5-yl)phenyl]methyl}cyclopropanamine
N2-benzyl-6-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-1,3,5-triazine-2,4-diamine
N4-methyl-N4-[3-(1-methyl-1H-imidazol-2-yl)propyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-hydroxypyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenylpyrimidine-5-carboxamide
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-methyl-5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyrimidin-2-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]acetamide
(3aS,6aR)-5-(5-chloropyridin-2-yl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-cyclooctyl-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
2-chloro-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]piperazine-1-sulfonamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-4-yl)propan-1-one
methyl 3-(4-fluorobenzenesulfonamido)-5-({[2-(methylsulfanyl)-1,3-thiazol-4-yl]formamido}methyl)benzoate
4'-[(3-methoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(2R,6R)-4-(dimethylcarbamoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-(diethylamino)ethan-1-one
3-{[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
3-(4-fluorophenyl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1H-pyrazole-5-carboxamide
4-{3-[(4,4-dimethylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}morpholine