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(1H-imidazol-2-ylmethyl)(methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
(3aS,6aS)-2-methanesulfonyl-5-(2-methylpyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-acetamido-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]acetamide
methyl 3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-amino-3-cyano-4-[5-(hydroxymethyl)furan-2-yl]-5H,6H-furo[2,3-h]quinoline-9-carboxylic acid
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
3-[3-(furan-2-yl)-5-[2-(methylamino)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-(furan-2-ylmethyl)-2-[5-oxo-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-[4-(4-fluorophenyl)piperazin-1-yl]-4-(pyridin-3-yl)pyrimidine
5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-(3-phenylpropyl)piperidin-2-one
1-[2-methyl-4-({3-[(5-methylpyridin-2-yl)amino]propyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)quinolin-2-amine
1-(furan-2-ylmethyl)-N-[1-(methylcarbamoyl)cyclohexyl]piperidine-3-carboxamide
3-(4-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenyl)prop-2-yn-1-ol
2-benzyl-5-formamido-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-{[(4-cyanopyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-benzyl-4-(4-methylpentyl)-1,4-diazepan-6-ol
(1S,9S)-11-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(2-methoxyphenyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(6-methylpyridin-3-yl)spiro[2.4]heptane-1-carboxamide
(2R)-N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-acetamidopropanamide
N-({1-[(2-hydroxyphenyl)methyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
3-(hydroxymethyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-ol
6-[(diethylamino)methyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
9-(2-chlorophenyl)-N,N,15-trimethyl-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-[(4aR,7aS)-4-[(3,5-difluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
4-(1H-imidazol-1-yl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}butan-1-one
{[5-(ethanesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5-methyl-1,3,4-oxadiazol-2-amine
2-oxo-N-propyl-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxamide
2-(2-chloro-6-methoxyphenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
1-(2-{[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)amino}ethyl)cyclopentan-1-ol
2-cyclopropyl-4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2,6-difluorophenyl)methyl](pyridin-3-ylmethyl)amine
N-[(1S)-1-[3-(5-chloro-2-methylphenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-imidazol-4-yl)ethyl]acetamide
{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-propanamidobenzamide
N-[(3R,4R)-1-[(4-chloro-3-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl]propanoate
4,6-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(5-ethylthiophene-2-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
3-{[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}-N-(3-fluorophenyl)propanamide
methyl 1-methyl-4-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)piperazine-2-carboxylate
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(pyridin-2-yl)acetamide
4-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
2-{2-[3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-8-methyl-2,8-diazaspiro[4.5]decan-3-one