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2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrophthalazin-1-one
(2S)-3-(4-hydroxyphenyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]formamido}propanoic acid
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(1-benzofuran-2-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)sulfamoyl}-N-ethyl-N-methylbenzamide
2-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)quinoline
4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-1-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl(pyrazin-2-ylmethyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-methyl-3-[methyl(pyridin-4-ylmethyl)amino]butanamide
3-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
2-[1-(3,4-difluorophenyl)-5-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl]acetamide
3-(5-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}thiophen-3-yl)prop-2-yn-1-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(4-phenylphenyl)methyl]pyrrolidine-2-carboxamide
(butan-2-yl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-2-chloro-6-methoxyphenol
3-phenyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazine
(1S,5R)-3-[4-(dimethylamino)benzoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-8-[(4-methyl-1H-imidazol-5-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethylamino)ethyl]-3-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-4-methoxybenzamide
3-(propan-2-yl)-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-methylbut-2-en-1-one
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
2,8-dimethyl-4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-propanamidobenzamide
1-(5-acetylpyridin-2-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-benzyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-sulfonamide
methyl 2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
{4-[(3-fluorophenyl)methyl]-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}methanol
5-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-phenyl-N-{1-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole
2-(1-tert-butyl-1H-pyrazol-4-yl)-6-ethyl-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-phenyl-1,2,4-oxadiazole
(2S)-2-[2-(3-chlorophenyl)-1H-imidazol-1-yl]-3-phenylpropanamide
1-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1,4-diazepane-6-carboxylic acid
3-({2-[(2S,4S)-4-amino-2-(ethylcarbamoyl)pyrrolidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
1-benzyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N'-cyclopentyl-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]ethanediamide
2-[4-({1-[2-(benzenesulfonyl)ethyl]-7-chloro-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
{[6-(cyclohexylmethoxy)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(pyridin-3-ylmethyl)amine
2-[4-(6-cyclopropylpyrimidin-4-yl)piperazin-1-yl]-4-methyl-6-(trifluoromethyl)pyrimidine
N-ethyl-N-[2-(phenylsulfanyl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-cyclopropyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,3,4-oxadiazol-2-amine
(2S,4R)-4-amino-N-(1-benzothiophen-5-ylmethyl)pyrrolidine-2-carboxamide
7-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-(4-chlorophenoxy)-N-[(3R)-piperidin-3-yl]piperidine-4-carboxamide
5-methyl-2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol