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{5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-2-ethoxyphenyl}methanol
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
propan-2-yl N-{[(3S,4S)-3-hydroxy-1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}carbamate
ethyl 4-({[7-fluoro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)piperidine-1-carboxylate
2-benzyl-9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-{[5-(3-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
4-{3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]propanamido}benzamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
8-(2-methoxybutanoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(3-methoxypiperidine-1-carbonyl)piperidin-1-yl]-4,6,7-trimethylquinazoline
4-{4-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
N-(1-ethyl-1H-indazol-3-yl)-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-1-(3-aminopropyl)-6-[4-(propan-2-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
(1S,4S)-2-(2,5-dimethoxyphenyl)-5-[(5-methylthiophen-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(3-chlorophenyl)-4-[3-(3-methoxyphenoxy)propyl]piperazin-2-one
6-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetate
N-(1-methoxypropan-2-yl)-3-azaspiro[5.5]undecan-9-amine
7-chloro-2-methyl-4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-7-[5-(propan-2-yl)thiophene-3-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-[(1-ethyl-1H-pyrazol-3-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
N-{3-[methyl(phenyl)amino]propyl}morpholine-2-carboxamide
(1R,3S)-3-methoxy-7-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-{[4-(dimethylamino)piperidin-1-yl]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[4-methyl-2-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrimidin-5-yl]ethan-1-one
(1R,3S)-1-hydroxy-3-methoxy-N-(2-methoxy-5-methylphenyl)-7-azaspiro[3.5]nonane-7-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-[benzyl(2-hydroxyethyl)amino]-1-[2-(piperidin-1-yl)ethyl]azepan-2-one
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-(pyridin-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-methyl-2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
5-methyl-1-[5-(2-methylpropanoyl)thiophen-2-yl]-1H-pyrazole-3-carboxylic acid
1-ethyl-8-[(3-methoxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(trifluoromethyl)benzamide
N-cyclohexyl-3-[(4-methyl-3-phenyl-1H-pyrazol-5-yl)formamido]propanamide
N-{[7-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
N-[2-(N-methylmethanesulfonamido)ethyl]-3-(1H-pyrazol-1-yl)benzamide
2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine-4-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[(1-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(5-methylhexan-2-yl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-{[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-6-methylquinolin-4-ol
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
4-(4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)butan-1-ol
8-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol