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ethyl 1-[2-(dimethylamino)ethyl]-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-amino-4-(5-fluoro-2-methoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-methylpyrido[2,3-d]pyrimidin-4-amine
1-(1-cyclopropylethyl)-5-(2-methoxynaphthalen-1-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl}acetamide
3-{[(4-chlorophenyl)methyl]({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino}propan-1-ol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-{4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]morpholin-3-yl}acetic acid
2-{[cyclopropyl(thiophen-3-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
N-benzyl-2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-sulfonamide
5-methanesulfonyl-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
(3aS,6aS)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydropyrrolo[2,3-c]pyrrole
(3aS,6aS)-2-[2-(4-chlorophenyl)acetyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(3R,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-(2H-1,3-benzodioxol-5-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
8-(6-aminopyrimidin-4-yl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-1-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-6-(3-methylphenyl)pyridine-3-carbonitrile
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]oxolane-2-carboxamide
N-[4-(methylamino)butyl]-1-[3-(1,3-oxazol-5-yl)phenyl]piperidin-4-amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1,4-diazepane
2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-methyl-2-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)propanamide
methyl (2R,4S)-4-hydroxy-1-(oxan-4-ylmethyl)piperidine-2-carboxylate
(2R,3R,6R)-5-(2,1,3-benzoxadiazol-4-ylmethyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-methoxyphenyl)-4-(3-phenylbutanoyl)piperazin-2-one
3-methoxy-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}propan-1-one
8-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
6-(2,5-dimethylfuran-3-yl)-2-{2-[(3-ethylmorpholin-4-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-{4-hydroxy-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-1-yl}-2-methylpropan-1-one
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyridine-4-carboxamide
2-(2-chloro-6-fluorophenyl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
2-benzyl-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-N-methylethane-1-sulfonamide
6,7-dimethyl-4-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]-2H-chromen-2-one
2-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,3-dihydro-1,2-benzothiazol-3-one
2-{1-methyl-5-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-(2-methoxyethyl)-4-methyl-3-[2-oxo-2-(piperidin-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-(quinolin-6-ylmethyl)pyrimidine-5-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
(3S,4R)-3-ethyl-4-methyl-1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperidin-4-ol
1-methyl-N-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
7-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-cyclopropyl-N-[1-(3-methylphenyl)piperidin-4-yl]-6-oxopiperidine-3-carboxamide
1-(4-{2-azaspiro[4.4]nonan-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-ethoxyethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-6-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide