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1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-[4-(3-fluorophenyl)phenyl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)piperidin-4-amine
2-methyl-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
methyl 3-[(3S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
dimethyl(3-{2-[1-(2,4,6-trimethylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
1-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1-benzothiophen-7-yl)-6-cyclobutyl-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1-methyl-1H-pyrazole-3-carbonyl)pyrrolidine-3-carboxylic acid
[(3R,5S)-1-[(2,3-dichlorophenyl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
4,4,4-trifluoro-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]butan-1-one
ethyl 1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
4-methoxy-3-(3-methylthiophen-2-yl)benzamide
{1-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methanol
8-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-2-yl)propan-1-ol
1-{[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,3-dimethylurea
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
2-{[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-4-methoxyphenol
4-(morpholine-4-carbonyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyridin-2-amine
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[2-(adamantan-1-ylsulfanyl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(1'-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
N-(oxolan-2-ylmethyl)-5-[1-(pyridin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidin-2-amine
4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
6-(2,1,3-benzothiadiazol-5-ylmethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]azetidin-3-yl}pyridine
[(4-methanesulfonylphenyl)methyl][(2-methylphenyl)methyl](2-methylpropyl)amine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidin-2-amine
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)propanamide
(3S)-N-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-amine
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-(1-methyl-1H-indazol-6-yl)piperidine-1-carboxamide
4-(azepane-1-carbonyl)-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
N-[1-(pyridin-3-yl)propan-2-yl]-3-(trifluoromethyl)benzamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(piperidin-1-ylmethyl)benzamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
1-phenyl-4-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperazine-2-carboxylic acid
1-(methoxymethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}cyclobutane-1-carboxamide
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-ethylpyridine-4-carboxamide
2-{[(1S,2S)-2-hydroxycyclohexyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-4-carboxamide
[5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)furan-2-yl]methanol
3-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methylphenol