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4-chloro-1-methyl-5-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-3-(trifluoromethyl)-1H-pyrazole
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(4-phenoxybenzoyl)piperidine
1-[(1S,5R)-6-(2-hydroxy-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(adamantan-2-ylmethyl)-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-N-(2-methoxyethyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(3-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-5-methyl-1,3-oxazole-4-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
2-amino-4-({[(2S)-1-ethylpyrrolidin-2-yl]methyl}amino)quinazoline-6-carboxylic acid
1-[(2-fluorophenyl)methyl]-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
1-(furan-2-ylmethyl)-N-(4H-1,2,4-triazol-4-yl)piperidine-3-carboxamide
(4aS,7aR)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[1-(quinolin-4-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-[(3-methylpyridin-4-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}benzamide
1-(2-methoxyphenyl)-3-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-(2-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)acetamide
4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-1-methylpiperidin-4-ol
2-(1-ethylpiperidin-4-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
(3aR,6aS)-5-(5-chloronaphthalene-1-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1,3-benzoxazol-2-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidin-4-amine
(1R,5S)-N-(2H-1,3-benzodioxol-5-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-{2-[methyl({[4-(trifluoromethoxy)phenyl]methyl})amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)-4-methylbenzamide
(3S,5R)-1-[2-(2-methylphenyl)acetyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
(3S,9aR)-3-(cyclohexylmethyl)-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(2S)-2-hydroxypropanoyl]-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-{[5-(1-methanesulfonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
(1S,4S)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,3,3-trimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
1-[(4-methoxy-2,5-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}butanamide
N-[(2,4-difluorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{[3-(furan-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
(3S,5R)-3-(hydroxymethyl)-N-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
1-{3-[3-cyclopentyl-1-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
7-cyclobutaneamido-N-(2,3-dihydro-1H-inden-1-yl)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
(4aS,8aR)-1-methanesulfonyl-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyridine-4-carbonitrile
(3S,4R)-4-(2-methoxyphenyl)-1-(4-methylpiperidine-4-carbonyl)pyrrolidine-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2,2-dimethylcyclopropane-1-carboxamide
4-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(piperidin-1-yl)piperidine
N-(4-fluoro-3-methoxyphenyl)-4-(thian-4-yl)piperazine-1-carboxamide