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2-[(3,5-difluorophenyl)methyl]-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-ethyl-9-(3-methylbenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
N4-methyl-N2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
5-[1-(diphenylmethyl)-1H-1,2,3-triazol-4-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
7-(cyclobutylmethyl)-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-(pyridin-4-ylsulfanyl)acetamide
7-[2-(phenylformamido)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(4-methyl-1,4-diazepan-1-yl)-N-[3-(pyridin-3-yl)propyl]acetamide
3-({4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}sulfonyl)pyridine
4-(8-methoxy-2H-chromen-3-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-ethyl-4-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)piperidine-1-carboxamide
2-methyl-4-{4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}-6-methoxyphenol
2-(2-hydroxyethyl)-9-(1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{3-[(2,4-difluorophenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-yl}methanol
(1R,7S)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide
8-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methoxypropanamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
3-fluoro-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methoxybenzamide
5-[4-(1-ethoxyethyl)phenyl]pyridine-2-carbonitrile
(4S)-3-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
4-(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)morpholine
(4aS,7aR)-1-(2-hydroxyacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]acetamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
3-methoxy-2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-4-oxobutane-1-sulfonamide
4-{[4-(2-methylphenyl)phenyl]methyl}-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(dimethyl-1,2-oxazol-4-yl)methyl]({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-{1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}acetamide
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
1-(oxolane-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(2,3-dimethylphenyl)methyl]-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aR)-6-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(3-fluorobenzoyl)-decahydro-1,6-naphthyridin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
methyl 3-cyclobutaneamido-5-{[(2,4-difluorophenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(3-chloro-4-propanamidophenyl)-N'-(2-ethylphenyl)ethanediamide
N-(cyclohex-1-en-1-ylmethyl)-3-fluoro-2-methoxybenzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(3-methylphenoxy)benzoyl]pyrrolidin-3-yl]methanol