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2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyridine-3-carbonitrile
3-[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-{[1-(azepan-1-yl)propan-2-yl]amino}ethyl)-N-methylmethanesulfonamide
3-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1'-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[3-(pyridin-3-yloxy)propyl]pyridin-2-amine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidine
N-[(3-chlorophenyl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-hydroxy-1-(2-methoxyethyl)-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2-dihydrophthalazin-1-one
ethyl 1-(2-carbamoylphenyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-[(1-methylpiperidin-3-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[furan-2-yl(phenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
4-(4-chlorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]butanamide
5-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-(methoxymethyl)thiophene-2-carboxamide
4-[2-(1H-imidazol-2-yl)benzoyl]-1-methylpiperazine-2-carboxylic acid
2-phenyl-N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
1-[(2S,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
1'-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-indole-6-carboxamide
N-[(2-methoxyphenyl)methyl]-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-[3,5-dimethyl-4-(quinolin-3-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
1-(4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)butan-1-ol
1-(4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole-3-carboxamide
2-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidin-1-yl}pyrimidine
2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
7-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]-1-[4-(2-fluorophenyl)piperazin-1-yl]propan-1-one
1-{5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
N,N-dimethyl-2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}-2-phenylacetamide
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{4H,5H,6H,7H,8H-cyclohepta[b]thiophen-2-ylformamido}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-[2-(2-ethylphenoxy)ethyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-methyl-4-[(4-methyl-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
2-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}pyridine
(3aR,7aS)-2-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]{[4-(methylsulfanyl)phenyl]methyl}amine
1-(2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}ethyl)piperidine-3-carboxamide