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4-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
6-(3,5-difluorophenyl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
5-(3-methylthiophen-2-yl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
8-(1-aminocyclopropanecarbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-methoxy-3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
2-[(cyclopropylmethyl)sulfanyl]-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-(3-hydroxypropyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N,N-dimethylpyridine-3-carboxamide
N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
2-(1-ethylpiperidin-3-yl)-7-methyl-1H-1,3-benzodiazole
5-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(4-methyl-2-oxo-2H-chromen-6-yl)oxy]propanamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-methanesulfonyl-4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepane
1-[(2-methoxyphenyl)methyl]-1-(3-methoxypropyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
4-[(2S)-2,3-dihydroxypropyl]-1-(2-methoxyphenyl)piperazin-2-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2,3-difluorobenzoyl)-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-acetyl-N-[(6-methylpyridin-2-yl)methyl]benzamide
1-{[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,4-triazole
3-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzoic acid
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N-methylpyrimidin-2-amine
1-{3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}azepan-2-one
N-[(4,6-dimethylpyridin-3-yl)methyl]-5-ethyl-2-methylpyrimidin-4-amine
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-1-[4-(4-fluorophenyl)piperazin-1-yl]ethan-1-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,N-diethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(3S,4R)-1-[(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
(1R,5R)-N-(2-chlorophenyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,4-diazepane
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(trifluoromethyl)morpholin-4-yl]acetamide
1,9-dimethyl-4-[4-(1H-pyrazol-1-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methylbenzamide
N-methyl-1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidine-3-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-N-(2,6-dimethylphenyl)piperidine-1-carboxamide
N-[(3S,4R)-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-methyl-N-(oxolan-2-ylmethyl)-2-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
5-(2-methylpropyl)-3-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
2-({2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridine-3-carboxylic acid
{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
1-(1,2-oxazol-3-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
2-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]morpholin-3-yl}acetic acid
N-[(3-ethoxyphenyl)methyl]-2-(2-oxopyrrolidin-1-yl)-N-(prop-2-en-1-yl)propanamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol