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(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-methoxyphenyl)-3-methyl-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
4-{4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
3-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
4-ethoxy-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine
N-methyl-3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
ethyl 3-{4-[1-(carbamoylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}benzoate
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[(3S)-2-oxoazepan-3-yl]piperidine-4-carboxamide
4-({5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-({[(3R,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(1-benzofuran-2-yl)-2-{[3-(dimethylamino)propyl](methyl)amino}acetic acid
N-cyclohexyl-1-ethyl-N-(2-hydroxy-2-phenylethyl)-1H-pyrazole-3-carboxamide
2-{2-[(3,4-dimethylpiperazin-1-yl)methyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
ethyl 4-{3-[benzyl(methyl)amino]piperidin-1-yl}piperidine-1-carboxylate
2-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
2-(1-benzyl-4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
ethyl 2-[(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)amino]acetate
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
9-(oxane-4-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N,4-dimethyl-2-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}aniline
1-(3-chloropyridin-2-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanamide
(1R,5R)-6-(1-benzofuran-5-ylmethyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-methylfuran-2-yl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,3S)-3-{[(8-methoxyquinolin-5-yl)methyl](methyl)carbamoyl}cyclopentane-1-carboxylic acid
1-ethyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2,3-dimethylphenoxy)ethan-1-one
1-methyl-3-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
5-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylpyridin-2-amine
(3S,4S)-1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
4-(4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)piperidin-4-ol
N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-methyl-N-(2-phenylethyl)piperidin-4-amine
1-[4-(4-methoxyphenoxy)phenyl]-3-(oxan-4-yl)urea
5-methyl-1-(2-oxo-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(furan-2-yl)ethane-1,2-dione
N-[(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]-4,4,4-trifluorobutanamide
methyl 3-(oxolane-2-amido)-1-(3-phenylpropyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]azepan-3-amine
2-[4-(1-methanesulfonylpyrrolidine-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-(1-cyanocyclohexyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-imidazol-4-ylmethyl)piperidin-3-ol
1'-(azepane-4-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-{2-[1-phenyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetamide
N-[2-(morpholin-4-yl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one