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(3aS,6aS)-2-(dimethylcarbamoyl)-5-(3-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aR,5S,6S,7aS)-2-(3-methyl-1H-pyrazole-5-carbonyl)-octahydro-1H-isoindole-5,6-diol
N-methyl-3-[N-methyl-1-(3-phenylphenyl)formamido]butanamide
1-[(2,2-dimethyloxan-4-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-[(4-methoxyphenyl)methyl]-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{2-[(4-benzylpiperidin-1-yl)methyl]-4-methoxyphenoxy}-3-(dimethylamino)propan-2-ol
1-(4-ethylpiperazin-1-yl)-3-[1-(4-phenylbutan-2-yl)piperidin-4-yl]propan-1-one
2-{[5-cyclohexyl-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1,4-diazepane
1-(4-{[2-(1H-pyrazol-4-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-(3-methanesulfonamidophenyl)-4-(pyrimidin-2-yl)piperazine-1-carboxamide
N-[(2,3-difluorophenyl)methyl]-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[1-(2-ethylpyrimidine-5-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-[2-(trifluoromethyl)benzoyl]piperidin-3-yl]methanol
1-(2,1,3-benzoxadiazol-4-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-methyl-4-[methyl({2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
2-({4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)pyrimidine
N-(1-methyl-2-oxopyrrolidin-3-yl)-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N,3,5-trimethyl-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-1H-indole-2-carboxamide
4-(3-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-4H-1,2,4-triazole
(1S,5R)-6-(cyclopropylmethyl)-3-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-N,N-diethyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N4-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N,N-dimethyl-5-{[(5-methylfuran-2-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-benzyl-3-[3-(thiophen-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(5-acetylthiophen-3-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N,N-dimethyl-5-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]pyridin-2-amine
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(1-methylpiperidin-4-yl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(2-methoxyethyl)-4-[5-(1,2-oxazol-3-yl)thiophen-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[1-(2-methoxyacetyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-2-methylquinoline
1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
3-(3-fluorophenyl)-4-[3-(methoxymethyl)benzoyl]piperazin-2-one
N-[2-(piperidin-1-ylmethyl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
2-benzyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]pyrimidine
5-(3-methoxyphenoxymethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
N'-(2-fluorophenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}ethanediamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-{1-methyl-4-[(trimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
propan-2-yl 2-chloro-5-({[2-(1H-imidazol-4-yl)ethyl]carbamoyl}amino)benzoate
1-{3-[({2-[3-(hydroxymethyl)piperidin-1-yl]-7-methoxyquinolin-3-yl}methyl)amino]propyl}pyrrolidin-2-one