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1-methyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2,4-difluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
2-{2-[(4-ethyl-1,4-diazepan-1-yl)methyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[2-(oxan-4-yl)ethyl]amine
2-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)ethan-1-ol
6-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-1,3-benzothiazole-6-carboxamide
1-(azepan-1-yl)-3-[4-({[(3-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxo-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
1-{4-[2-methoxy-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-(2,4-difluorophenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(3,4-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-[methyl({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl})amino]propan-1-ol
N-(oxan-4-ylmethyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
N-[2-(2-ethoxyphenyl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
4-hydroxy-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-(2-cyclopropylacetyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
7-{[4-(2-methylpropyl)phenyl]methyl}-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(2-fluorophenyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1H-pyrazole-5-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2R)-1-hydroxybutan-2-yl]pyrimidine-5-carboxamide
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
3-benzyl-5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
2-amino-4-(4-methanesulfonylphenyl)-6-(4-methoxyphenyl)pyridine-3-carbonitrile
2-methyl-1-(2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1H-indole-3-carbonitrile
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(4-fluorophenoxy)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
N-(3,5-dimethoxyphenyl)-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
4-{4-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[2-(pyridin-2-yl)ethyl]benzamide
(1R,3S)-7-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
1-(3-fluoropyridin-4-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
2-[4-(4,6-dimethoxypyrimidin-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
1-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
2-methoxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-4-carboxamide
2-{[3-(1H-imidazol-1-yl)propyl]amino}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
4-(5-{1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-imidazol-2-yl}-1,3-thiazol-2-yl)morpholine
3-({[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
2-[9-(3-methyl-1H-pyrazole-5-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N6-(3-methoxypropyl)-N5-methyl-N5-(quinolin-5-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-{1-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]pentyl}pyridine
1-(butan-2-yl)-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
2-cyclopropyl-5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
1-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol