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N5-cycloheptyl-N3-methyl-4-oxo-1-(propan-2-yl)-N3-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
7-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(oxan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
2-(5-acetylthiophen-3-yl)-N-(furan-2-ylmethyl)acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyrimidin-2-yl)piperidin-3-ol
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
(2R,6R)-4-[5-(methoxymethyl)furan-2-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(1-phenyl-1H-pyrazol-5-yl)-2-[3-(pyridin-4-yl)-1H-indazol-1-yl]acetamide
(2S,4S)-4-[(adamantan-2-yl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-{2,7-diazaspiro[4.5]decan-7-yl}-3-(2-hydroxyphenyl)propan-1-one
(2S)-1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxamide
[(3R,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-methoxy-N-{[3-(methylsulfanyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
7-(1,3-benzothiazol-2-yl)-4-(oxolan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
7-chloro-N-(3-phenyl-1,2,4-thiadiazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
1-{3-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]phenyl}ethan-1-one
methyl (2S)-1-[2-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
(2S,4R)-4-amino-N,N-diethyl-1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
5-{4-[2-(2-aminoethyl)quinazolin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-(1H-imidazol-4-ylmethyl)-4-(oxane-4-carbonyl)-1,4-diazepan-6-ol
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]azonane
1-[2-(propan-2-yl)pyrimidine-4-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methyl-4-{4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
1-{1-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]cyclohexyl}piperidine
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(pyridin-4-yl)-1H-indazol-1-yl]acetamide
(3R,4R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-cyclohexyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(1-phenyl-1H-pyrazol-5-yl)urea
methyl 1-[(3R,5S)-1-(cyclohexylmethyl)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[1-(cyclohexylmethyl)-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
1-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
methyl 3-benzamido-5-{[(4-methylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
dimethyl[1-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]amine
4-benzyl-3-ethyl-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,4-diazepan-5-one
4-[1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]benzoic acid
N-[2-(2-ethoxyphenoxy)ethyl]-3-methoxy-N,2,2-trimethylpropanamide
2-(4-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-[4-(2-fluorophenoxy)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
(2E)-3-(2-chlorophenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)prop-2-enamide
4-{[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1,2-oxazole
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
2-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-3,5,6-trimethylpyrazine
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
7-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one