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N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]-2-(4-ethylpiperazin-1-yl)acetamide
3-(methanesulfonylmethyl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine
methyl({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-N-(3-fluorophenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one
8-[8-(trifluoromethyl)quinolin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
6-chloro-N-[(3-propyl-1,2-oxazol-5-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
N-[(1R,3R)-3-aminocyclopentyl]-2-hydroxynaphthalene-1-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
7-(2-hydroxyethyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[5-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
4-(6-aminopyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-3-(pyrrolidin-1-yl)propan-2-ol
N-[(3S,4R)-1-[4-(carbamoylamino)benzenesulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-(2-methoxyethoxy)-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
(1S,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-[4-(5-methoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
2,9-dimethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-1'-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(5S)-5-{3-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-[5-(methoxymethyl)furan-2-carbonyl]azocane
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-methyl-4-{[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(4-methylphenyl)cyclopropane-1-carboxamide
5-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(1-acetylpiperidin-4-yl)-5-methyl-5-phenylpiperidin-2-one
2-(4-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
[2-(1H-imidazol-1-yl)ethyl][(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]methylamine
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(methylamino)ethan-1-one
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
5-[({[3-(2-{4-[2-(4-fluorophenyl)acetyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-ethyl-4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-N'-(4-methylphenyl)propanediamide
1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
9-(7-chloroquinolin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{[1-(4-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-[3-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methyl-1H-indazole
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
2-(3-hydroxypropyl)-9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2,3-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
1-(3-chlorophenyl)-5-oxo-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]pyrrolidine-3-carboxamide