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2-{4-[6-amino-5-cyano-4-(5-methylfuran-2-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
N2,N2,N4,N4-tetramethyl-7-(pyrrolidine-1-sulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
8-fluoro-N-[(2R)-1-hydroxybutan-2-yl]quinoline-2-carboxamide
(5-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-2-methoxyphenyl)methanol
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
1-{4-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenyl}imidazolidin-2-one
6-fluoro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperazine-1-carbaldehyde
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(methoxymethyl)thiophene-2-carboxamide
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(methoxymethyl)piperidine
3-[(2R,3R,6R)-5-[(2-fluoro-5-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-(1H-1,2,4-triazol-3-yl)urea
3-(1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)piperidine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
2-[(2,3-dihydro-1-benzothiophen-2-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)benzonitrile
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
4-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}sulfonyl)benzonitrile
1-(2-ethoxyethyl)-5-(1,4-oxazepane-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N,N,5-trimethyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(4-methoxyphenyl)methyl]piperidine
(1H-imidazol-2-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
5-(2-chloro-4-fluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
4-[1-(3-ethoxybenzoyl)piperidin-3-yl]benzoic acid
1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,5R)-N,N-dimethyl-6-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1,2-oxazol-3-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}sulfonyl)morpholine
5-(1H-1,3-benzodiazole-5-carbonyl)-1-benzyl-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4S)-1-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(2-{[4-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
1-(azocan-1-yl)-3-[2-methoxy-5-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
(3R,9aR)-8-(4-chlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-chloro-N-{2-[(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]ethyl}benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
6-[4-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
1-benzyl-3-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]urea
1-(4-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
3-(4-hydroxyphenyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-pyrazole-5-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
7-(2-methylphenyl)-4-(1-methylpyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
9-(1-ethylpiperidine-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
4-{1-ethyl-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazol-3-yl}benzamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-4-(1H-pyrrol-1-yl)phenol