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N-(2H-1,3-benzodioxol-5-yl)-1-[(6-chloroquinolin-2-yl)methyl]piperidin-3-amine
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-ethyl-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
8-chloro-N-(cyclobutylmethyl)-2-methyl-N-(oxolan-2-ylmethyl)quinoline-4-carboxamide
2-(methylsulfanyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-{2-cyclobutyl-1-methyl-7-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
4,6-dimethyl-5-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-(naphthalen-1-ylmethyl)morpholine
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-[2-(1H-imidazol-4-yl)acetyl]pyrrolidine-2-carboxamide
3-(4-cyclopropanecarbonyl-3-fluorophenyl)-5-methylpyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(pyridin-3-ylmethyl)acetamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
(2S,4S)-4-[4-(4-cyanobenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N,N-dimethyl-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-1H-pyrrole-2-carboxamide
1-(furan-2-yl)-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethane-1,2-dione
1-[1-(propan-2-yl)piperidine-3-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-butyl-N-[(2-fluorophenyl)methyl]but-3-enamide
3,5-dimethyl-1-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
1-(4-{7-chloro-3-[({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}amino)methyl]quinolin-2-yl}piperazin-1-yl)ethan-1-one
7-cyclopentyl-2-[2-(1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-methoxyphenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclopentane-1-carboxamide
3-(2-ethylbutyl)-8-(2-methyl-1,3-thiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3-fluorophenyl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
3-(2-methoxyphenoxy)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidine
(2S,4R)-4-(dimethylamino)-1-[(3-ethoxy-2-hydroxyphenyl)methyl]pyrrolidine-2-carboxylic acid
4-{4-[(2,2-dimethyloxan-4-yl)methyl]piperazin-1-yl}benzoic acid
2-{4-[(2E)-3-phenylprop-2-en-1-yl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
(3R,4R)-3-cyclobutyl-1-(4-methanesulfonylbenzoyl)-4-methylpyrrolidin-3-ol
5-oxo-1-phenyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2,5-dihydro-1H-pyrazole-3-carboxamide
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(4-chlorophenyl)morpholine
2-(2-methoxyethyl)-8-(2-phenoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
7-methoxy-3-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-[2-chloro-5-(trifluoromethoxy)phenyl]-N,N-dimethylbenzamide
(3aS,6aS)-2-cyclohexyl-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-chloro-5-fluorophenyl)-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methylurea
2,5-dimethyl-N-[2-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[1-(2,4-dimethylbenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
5-(5-ethylfuran-2-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
5-methoxy-1-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-indole-2-carboxamide
3-[1-(4-hydroxy-3-methoxyphenyl)-N-methylformamido]-N-methylbutanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
5-(propan-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-oxazole-3-carboxamide
1-(4-chlorophenyl)-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
2-(4-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}piperidin-1-yl)acetamide