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1-tert-butyl-N-[(3-chloro-4-fluorophenyl)methyl]-5-oxopyrrolidine-3-carboxamide
methyl[(2-methylpyridin-4-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
6-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-1,3-benzoxazole
6-{4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
3-[2-(2-fluorophenyl)ethyl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-(propan-2-yl)-5-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole
4-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
1-[(4-chlorophenyl)methyl]-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
1,9-dimethyl-4-(1,2-oxazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N,N-diethylpropanamide
4-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine-4-carbonyl]morpholine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(propan-2-yloxy)ethyl]piperidine-4-carboxamide
3-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}azetidin-3-yl)pyridine
4-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
1-(2-cyclobutylacetyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-amino-3-ethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[4-(pyrimidin-2-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-ethyl-2-(morpholin-4-yl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-5-[(1-hydroxy-2-methylpropan-2-yl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-ol
ethyl 3,5-dimethyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrrole-2-carboxylate
2-(pyridin-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-6-methylpyridine
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3-(2-methylphenyl)propan-1-one
3-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)methyl]-1,2,3-oxadiazol-3-ium-5-olate
methyl 5-[(4-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methylbut-2-enamide
6-(1-phenoxyethyl)-2-[3-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-(2-methoxyphenyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazole-5-carboxamide
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
1-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrrolidine-3-carboxamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-{4-[4-(aminomethyl)piperidin-1-yl]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(1,3-thiazol-2-yl)acetamide
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
(1S,5R)-3-benzoyl-6-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-[(5-{[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]methyl}pyrimidin-2-yl)amino]acetic acid
(2S)-2-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidine-1-carboxamide
7-[cyclohexyl(methoxy)methyl]-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2,3-dihydro-1H-inden-2-yl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-benzyl-N,5-dimethyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(2S)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methanol
(2S,4S)-N,N-diethyl-1-methyl-4-(2-methyl-1-benzofuran-5-amido)pyrrolidine-2-carboxamide
1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
2-hydroxy-4-methyl-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]pentan-1-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
6,7-dimethoxy-2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-[1'-(5-fluoropyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[(2-ethoxypyridin-3-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid